ATE250597T1 - N-benzolsulfonyl-l-prolin derivate, verfahren zu ihrer herstellung und ihre therapeutische verwendung - Google Patents

N-benzolsulfonyl-l-prolin derivate, verfahren zu ihrer herstellung und ihre therapeutische verwendung

Info

Publication number
ATE250597T1
ATE250597T1 AT97945928T AT97945928T ATE250597T1 AT E250597 T1 ATE250597 T1 AT E250597T1 AT 97945928 T AT97945928 T AT 97945928T AT 97945928 T AT97945928 T AT 97945928T AT E250597 T1 ATE250597 T1 AT E250597T1
Authority
AT
Austria
Prior art keywords
group
pct
date
benzenesulfonyl
production
Prior art date
Application number
AT97945928T
Other languages
English (en)
Inventor
Pierre Dodey
Michel Bondoux
Khan Ou
Martine Barth
Patrick Houziaux
Original Assignee
Fournier Ind & Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fournier Ind & Sante filed Critical Fournier Ind & Sante
Application granted granted Critical
Publication of ATE250597T1 publication Critical patent/ATE250597T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT97945928T 1996-12-04 1997-11-14 N-benzolsulfonyl-l-prolin derivate, verfahren zu ihrer herstellung und ihre therapeutische verwendung ATE250597T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9614891A FR2756562B1 (fr) 1996-12-04 1996-12-04 Nouveaux composes de n-benzenesulfonyl-l-proline, procede de preparation et utilisation en therapeutique
PCT/FR1997/002049 WO1998024783A1 (fr) 1996-12-04 1997-11-14 Nouveaux composes de n-benzenesulfonyl-l-proline, procede de preparation et utilisation en therapeutique

Publications (1)

Publication Number Publication Date
ATE250597T1 true ATE250597T1 (de) 2003-10-15

Family

ID=9498333

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97945928T ATE250597T1 (de) 1996-12-04 1997-11-14 N-benzolsulfonyl-l-prolin derivate, verfahren zu ihrer herstellung und ihre therapeutische verwendung

Country Status (14)

Country Link
US (1) US6063791A (de)
EP (1) EP0944618B1 (de)
JP (1) JP4229219B2 (de)
AT (1) ATE250597T1 (de)
AU (1) AU5125798A (de)
CA (1) CA2273894C (de)
DE (1) DE69725167T2 (de)
DK (1) DK0944618T3 (de)
ES (1) ES2207752T3 (de)
FR (1) FR2756562B1 (de)
PL (1) PL186648B1 (de)
PT (1) PT944618E (de)
TR (1) TR199901242T2 (de)
WO (1) WO1998024783A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2790260B1 (fr) * 1999-02-26 2001-05-04 Fournier Ind & Sante Nouveaux composes de n-(benzenesulfonamide), procede de preparation et utilisation en therapeutique
CA2364178C (en) * 2000-12-05 2006-01-10 Yasuhiro Katsu N-benzenesulfonyl l-proline compounds as bradykinin antagonists
FR2819254B1 (fr) * 2001-01-08 2003-04-18 Fournier Lab Sa Nouveaux composes de la n-(phenylsulfonyl) glycine, leur procede de preparation et leur utilisation pour obtenir des compostions pharmaceutiques
ITMI20021247A1 (it) * 2002-06-07 2003-12-09 Menarini Ricerche Spa Antagonisti basici non peptidici della bradichinina e loro impiego informulazioni farmaceutiche
FR2840897B1 (fr) 2002-06-14 2004-09-10 Fournier Lab Sa Nouveaux derives d'arylsulfonamides et leur utilisation en therapeutique
US7080112B2 (en) * 2002-11-13 2006-07-18 International Business Machines Corporation Method and apparatus for computing an approximation to the reciprocal of a floating point number in IEEE format
SI1606288T1 (sl) 2003-03-25 2009-10-31 Fournier Lab Sa Derivati benzensulfonamida, postopek za njihovo pripravo in njihova uporaba za zdravljenje bolečine

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3617183A1 (de) * 1985-11-16 1987-05-27 Bayer Ag Substituierte benzylether
DE3632329A1 (de) * 1986-09-24 1988-03-31 Bayer Ag Substituierte phenylsulfonamide
AU686115B2 (en) * 1992-11-02 1998-02-05 Fujisawa Pharmaceutical Co., Ltd. Imidazo (I,2-a) pyridine derivatives as bradykinin antagonists, pharmaceuticals and processes for their preparation
AU680870B2 (en) * 1993-04-28 1997-08-14 Astellas Pharma Inc. New heterocyclic compounds

Also Published As

Publication number Publication date
JP4229219B2 (ja) 2009-02-25
DE69725167T2 (de) 2004-06-09
EP0944618B1 (de) 2003-09-24
WO1998024783A1 (fr) 1998-06-11
AU5125798A (en) 1998-06-29
DK0944618T3 (da) 2004-02-02
EP0944618A1 (de) 1999-09-29
PL186648B1 (pl) 2004-02-27
FR2756562A1 (fr) 1998-06-05
TR199901242T2 (xx) 1999-10-21
DE69725167D1 (de) 2003-10-30
ES2207752T3 (es) 2004-06-01
FR2756562B1 (fr) 1999-01-08
US6063791A (en) 2000-05-16
PT944618E (pt) 2004-02-27
CA2273894A1 (en) 1998-06-11
JP2001504854A (ja) 2001-04-10
PL334088A1 (en) 2000-01-31
CA2273894C (en) 2005-04-19

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