ATE415966T1 - Substituierte 3-amino-thieno(2,3-b)pyridine-2- amide und herstellungsverfahren sowie deren verwendung - Google Patents

Substituierte 3-amino-thieno(2,3-b)pyridine-2- amide und herstellungsverfahren sowie deren verwendung

Info

Publication number: ATE415966T1
Authority: AT; Austria
Prior art keywords: thieno; amides; pyridine; amino; substituted
Prior art date: 2002-06-06

Application number

AT03736796T

Other languages

English (en)

Inventor

Ch L Cywin

Z Chen

Jonathan Emeigh

R W Fleck

M Hao

E Hickey

W Liu

D R Marshall

Tina M Morwick

P Nemoto

R J Sorcek

S Sun

J Wu

Original Assignee

Boehringer Ingelheim Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-06-06

Filing date

2003-06-03

Publication date

2008-12-15

2003-06-03 Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma

2008-12-15 Application granted granted Critical

2008-12-15 Publication of ATE415966T1 publication Critical patent/ATE415966T1/de

Links

238000004519 manufacturing process Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
- C08G63/00—Macromolecular compounds obtained by reactions forming a carboxylic ester link in the main chain of the macromolecule
- C08G63/68—Polyesters containing atoms other than carbon, hydrogen and oxygen
- C08G63/695—Polyesters containing atoms other than carbon, hydrogen and oxygen containing silicon
- C08G63/6954—Polyesters containing atoms other than carbon, hydrogen and oxygen containing silicon derived from polxycarboxylic acids and polyhydroxy compounds
- C08G63/6956—Dicarboxylic acids and dihydroxy compounds
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
- C08G63/00—Macromolecular compounds obtained by reactions forming a carboxylic ester link in the main chain of the macromolecule
- C08G63/91—Polymers modified by chemical after-treatment
- C08G63/914—Polymers modified by chemical after-treatment derived from polycarboxylic acids and polyhydroxy compounds
- C08G63/916—Dicarboxylic acids and dihydroxy compounds

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Immunology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Polymers & Plastics (AREA)
Epidemiology (AREA)
Dermatology (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Toxicology (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Hematology (AREA)
Orthopedic Medicine & Surgery (AREA)
Transplantation (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Emergency Medicine (AREA)
Obesity (AREA)
Vascular Medicine (AREA)
Oncology (AREA)

AT03736796T 2002-06-06 2003-06-03 Substituierte 3-amino-thieno(2,3-b)pyridine-2- amide und herstellungsverfahren sowie deren verwendung ATE415966T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US38631202P	2002-06-06	2002-06-06
US45786703P	2003-03-26	2003-03-26

Publications (1)

Publication Number	Publication Date
ATE415966T1 true ATE415966T1 (de)	2008-12-15

Family

ID=29739900

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03736796T ATE415966T1 (de)	2002-06-06	2003-06-03	Substituierte 3-amino-thieno(2,3-b)pyridine-2- amide und herstellungsverfahren sowie deren verwendung

Country Status (26)

Country	Link
US (2)	US6964956B2 (de)
EP (2)	EP2008654A1 (de)
JP (2)	JP4364120B2 (de)
KR (1)	KR20050005548A (de)
CN (1)	CN100386329C (de)
AR (1)	AR040250A1 (de)
AT (1)	ATE415966T1 (de)
AU (1)	AU2003237330A1 (de)
BR (1)	BR0311605A (de)
CA (1)	CA2483890C (de)
DE (1)	DE60325051D1 (de)
DK (1)	DK1513516T3 (de)
EA (1)	EA008706B1 (de)
ES (1)	ES2318141T3 (de)
HR (1)	HRP20041154A2 (de)
IL (1)	IL164597A0 (de)
ME (2)	ME00355B (de)
MX (1)	MXPA04011246A (de)
NO (1)	NO20044599L (de)
NZ (1)	NZ537394A (de)
PE (1)	PE20040539A1 (de)
PL (1)	PL373424A1 (de)
RS (1)	RS105204A (de)
TW (1)	TWI296927B (de)
UY (1)	UY27834A1 (de)
WO (1)	WO2003103661A1 (de)

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2003
- 2003-06-03 DE DE60325051T patent/DE60325051D1/de not_active Expired - Lifetime
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- 2003-06-03 WO PCT/US2003/017343 patent/WO2003103661A1/en not_active Ceased
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- 2003-06-03 EP EP08164478A patent/EP2008654A1/de not_active Withdrawn
- 2003-06-03 KR KR10-2004-7019850A patent/KR20050005548A/ko not_active Ceased
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2004
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2005
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Publication number	Publication date
EA200401541A1 (ru)	2005-06-30
JP2005530816A (ja)	2005-10-13
UY27834A1 (es)	2003-12-31
EP1513516A1 (de)	2005-03-16
JP4364120B2 (ja)	2009-11-11
EA008706B1 (ru)	2007-06-29
ES2318141T3 (es)	2009-05-01
HRP20041154A2 (en)	2005-06-30
DE60325051D1 (de)	2009-01-15
ME00355B (me)	2010-06-30
EP2008654A1 (de)	2008-12-31
PE20040539A1 (es)	2004-10-21
MXPA04011246A (es)	2005-06-03
NO20044599L (no)	2005-02-16
AU2003237330A1 (en)	2003-12-22
IL164597A0 (en)	2005-12-18
NZ537394A (en)	2006-12-22
KR20050005548A (ko)	2005-01-13
JP2009102447A (ja)	2009-05-14
CA2483890C (en)	2012-12-11
US6964956B2 (en)	2005-11-15
EP1513516B1 (de)	2008-12-03
RS105204A (sr)	2006-12-15
BR0311605A (pt)	2005-02-22
US7405225B2 (en)	2008-07-29
AR040250A1 (es)	2005-03-23
CN100386329C (zh)	2008-05-07
US20040053957A1 (en)	2004-03-18
DK1513516T3 (da)	2009-10-19
MEP53508A (en)	2011-05-10
WO2003103661A1 (en)	2003-12-18
CN1649581A (zh)	2005-08-03
CA2483890A1 (en)	2003-12-18
TW200401640A (en)	2004-02-01
US20050288285A1 (en)	2005-12-29
PL373424A1 (en)	2005-08-22
TWI296927B (en)	2008-05-21
HK1080737A1 (zh)	2006-05-04

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