NO20044599L - 3-amino-tieno[2,3-b]pyridin-2-karboksysyreamid-forbindelser og fremgangsmater for fremstilling og anvendelser av dem - Google Patents

3-amino-tieno[2,3-b]pyridin-2-karboksysyreamid-forbindelser og fremgangsmater for fremstilling og anvendelser av dem

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Publication number
NO20044599L
NO20044599L NO20044599A NO20044599A NO20044599L NO 20044599 L NO20044599 L NO 20044599L NO 20044599 A NO20044599 A NO 20044599A NO 20044599 A NO20044599 A NO 20044599A NO 20044599 L NO20044599 L NO 20044599L
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NO
Norway
Prior art keywords
processes
preparation
thieno
pyridine
amino
Prior art date
Application number
NO20044599A
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English (en)
Inventor
Jiang-Ping Wu
Eugene Richard Hickey
Sanxing Sun
Tina Marie Morwick
Charles Cywin
Zhidong Chen
Jonathan Emeigh
Roman Wolfgang Fleck
Ming Hong Hao
Will Weimin Liu
Daniel R Marshall
Peter Nemoto
Ronald J Sorcek
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of NO20044599L publication Critical patent/NO20044599L/no

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Abstract

Beskrevet er forbindelser med formel (I), hvor R1 og R2 er definert her, som er anvendelige som inhibitorer av kinaseaktiviteten til IkB kinase(IKK)komplekset. Forbindelsene er derfor anvendelige ved behandling av IKK-medierte sykdommer omfattende autoimmune sykdommer, inflammatoriske sykdommer og kreft. Beskrevet er også farmasøytiske preparater omfattende disse forbindelser og fremgangsmåter for fremstilling av disse.
NO20044599A 2002-06-06 2004-10-25 3-amino-tieno[2,3-b]pyridin-2-karboksysyreamid-forbindelser og fremgangsmater for fremstilling og anvendelser av dem NO20044599L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38631202P 2002-06-06 2002-06-06
US45786703P 2003-03-26 2003-03-26
PCT/US2003/017343 WO2003103661A1 (en) 2002-06-06 2003-06-03 SUBSTITUTED 3-AMINO-THIENO[2,3-b]PYRIDINE-2-CARBOXYLIC ACID AMIDE COMPOUNDS AND PROCESSES FOR PREPARING AND THEIR USES

Publications (1)

Publication Number Publication Date
NO20044599L true NO20044599L (no) 2005-02-16

Family

ID=29739900

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NO20044599A NO20044599L (no) 2002-06-06 2004-10-25 3-amino-tieno[2,3-b]pyridin-2-karboksysyreamid-forbindelser og fremgangsmater for fremstilling og anvendelser av dem

Country Status (26)

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US (2) US6964956B2 (no)
EP (2) EP1513516B1 (no)
JP (2) JP4364120B2 (no)
KR (1) KR20050005548A (no)
CN (1) CN100386329C (no)
AR (1) AR040250A1 (no)
AT (1) ATE415966T1 (no)
AU (1) AU2003237330A1 (no)
BR (1) BR0311605A (no)
CA (1) CA2483890C (no)
DE (1) DE60325051D1 (no)
DK (1) DK1513516T3 (no)
EA (1) EA008706B1 (no)
ES (1) ES2318141T3 (no)
HR (1) HRP20041154A2 (no)
IL (1) IL164597A0 (no)
ME (2) ME00355B (no)
MX (1) MXPA04011246A (no)
NO (1) NO20044599L (no)
NZ (1) NZ537394A (no)
PE (1) PE20040539A1 (no)
PL (1) PL373424A1 (no)
RS (1) RS105204A (no)
TW (1) TWI296927B (no)
UY (1) UY27834A1 (no)
WO (1) WO2003103661A1 (no)

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