BRPI0606145A8 - Formas farmacêuticas sólidas de cloridrato de oxicodonaresistentes ao rompimento com liberação sustentada - Google Patents

Formas farmacêuticas sólidas de cloridrato de oxicodonaresistentes ao rompimento com liberação sustentada

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Publication number
BRPI0606145A8
BRPI0606145A8 BRPI0606145A BRPI0606145A BRPI0606145A8 BR PI0606145 A8 BRPI0606145 A8 BR PI0606145A8 BR PI0606145 A BRPI0606145 A BR PI0606145A BR PI0606145 A BRPI0606145 A BR PI0606145A BR PI0606145 A8 BRPI0606145 A8 BR PI0606145A8
Authority
BR
Brazil
Prior art keywords
sustained release
breakage
resistant
oxicodona
hydrochlorite
Prior art date
Application number
BRPI0606145A
Other languages
English (en)
Inventor
Judy Ashworth
Elisabeth Arkenau-Maric
Johannes Bartholomäus
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36384542&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0606145(A8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of BRPI0606145A2 publication Critical patent/BRPI0606145A2/pt
Publication of BRPI0606145A8 publication Critical patent/BRPI0606145A8/pt
Publication of BRPI0606145B1 publication Critical patent/BRPI0606145B1/pt
Publication of BRPI0606145B8 publication Critical patent/BRPI0606145B8/pt
Publication of BRPI0606145C1 publication Critical patent/BRPI0606145C1/pt

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    • B29C2793/009—Shaping techniques involving a cutting or machining operation after shaping
    • B—PERFORMING OPERATIONS; TRANSPORTING
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    • B29C35/00—Heating, cooling or curing, e.g. crosslinking or vulcanising; Apparatus therefor
    • B29C35/02—Heating or curing, e.g. crosslinking or vulcanizing during moulding, e.g. in a mould
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    • B29C43/00—Compression moulding, i.e. applying external pressure to flow the moulding material; Apparatus therefor
    • B29C43/22—Compression moulding, i.e. applying external pressure to flow the moulding material; Apparatus therefor of articles of indefinite length
    • B29C43/24—Calendering
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
    • B29C—SHAPING OR JOINING OF PLASTICS; SHAPING OF MATERIAL IN A PLASTIC STATE, NOT OTHERWISE PROVIDED FOR; AFTER-TREATMENT OF THE SHAPED PRODUCTS, e.g. REPAIRING
    • B29C45/00—Injection moulding, i.e. forcing the required volume of moulding material through a nozzle into a closed mould; Apparatus therefor
    • B29C45/0001—Injection moulding, i.e. forcing the required volume of moulding material through a nozzle into a closed mould; Apparatus therefor characterised by the choice of material
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    • B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
    • B29K2105/0005—Condition, form or state of moulded material or of the material to be shaped containing compounding ingredients
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    • B—PERFORMING OPERATIONS; TRANSPORTING
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    • B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
    • B29K2105/0005—Condition, form or state of moulded material or of the material to be shaped containing compounding ingredients
    • B29K2105/0044—Stabilisers, e.g. against oxydation, light or heat
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
    • B29K—INDEXING SCHEME ASSOCIATED WITH SUBCLASSES B29B, B29C OR B29D, RELATING TO MOULDING MATERIALS OR TO MATERIALS FOR MOULDS, REINFORCEMENTS, FILLERS OR PREFORMED PARTS, e.g. INSERTS
    • B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
    • B29K2105/25—Solid
    • B29K2105/251—Particles, powder or granules
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
    • B29K—INDEXING SCHEME ASSOCIATED WITH SUBCLASSES B29B, B29C OR B29D, RELATING TO MOULDING MATERIALS OR TO MATERIALS FOR MOULDS, REINFORCEMENTS, FILLERS OR PREFORMED PARTS, e.g. INSERTS
    • B29K2995/00—Properties of moulding materials, reinforcements, fillers, preformed parts or moulds
    • B29K2995/0037—Other properties
    • B29K2995/0056—Biocompatible, e.g. biopolymers or bioelastomers
    • B—PERFORMING OPERATIONS; TRANSPORTING
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    • B29L—INDEXING SCHEME ASSOCIATED WITH SUBCLASS B29C, RELATING TO PARTICULAR ARTICLES
    • B29L2031/00—Other particular articles
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    • B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
    • B29L—INDEXING SCHEME ASSOCIATED WITH SUBCLASS B29C, RELATING TO PARTICULAR ARTICLES
    • B29L2031/00—Other particular articles
    • B29L2031/772—Articles characterised by their shape and not otherwise provided for

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Abstract

FORMAS FARMACÊUTICAS RESISTENTES AO ROMPIMENTO COM LIBERAÇÃO SUSTENTADA. A invenção refere-se a uma forma farmacêutica que compreende uma substância fisiologicamente eficaz (A) com liberação pelo menos parcialmente sustentada, conforme o caso, um ou vários adjuvantes (B) fisiologicamente compatíveis e um polímero sintético ou natural (e), apresentando a forma farmacêutica uma resistência ao rompimento de pelo menos 400 N.
BRPI0606145A 2005-02-04 2006-02-06 formas farmacêuticas sólidas de cloridrato de oxicodona resistentes ao rompimento com liberação sustentada BRPI0606145C1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102005005446.3 2005-02-04
DE102005005446A DE102005005446A1 (de) 2005-02-04 2005-02-04 Bruchfeste Darreichungsformen mit retardierter Freisetzung
PCT/EP2006/001027 WO2006082099A1 (de) 2005-02-04 2006-02-06 Bruchfeste darreichungsformen mit retardierter freisetzung

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BRPI0606145A2 BRPI0606145A2 (pt) 2009-06-02
BRPI0606145A8 true BRPI0606145A8 (pt) 2018-05-29
BRPI0606145B1 BRPI0606145B1 (pt) 2019-09-17
BRPI0606145B8 BRPI0606145B8 (pt) 2019-11-05
BRPI0606145C1 BRPI0606145C1 (pt) 2021-05-25

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BRPI0606145A BRPI0606145C1 (pt) 2005-02-04 2006-02-06 formas farmacêuticas sólidas de cloridrato de oxicodona resistentes ao rompimento com liberação sustentada

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AR (2) AR054328A1 (pt)
AU (1) AU2006210145B9 (pt)
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