FI120586B - Menetelmä PTH:n ja PTHRP:n analogien valmistamiseksi, ja niiden käyttö osteoporoosin hoitoon - Google Patents

Menetelmä PTH:n ja PTHRP:n analogien valmistamiseksi, ja niiden käyttö osteoporoosin hoitoon Download PDF

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Publication number
FI120586B
FI120586B FI950169A FI950169A FI120586B FI 120586 B FI120586 B FI 120586B FI 950169 A FI950169 A FI 950169A FI 950169 A FI950169 A FI 950169A FI 120586 B FI120586 B FI 120586B
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glu
arg
lys
ser
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FI950169A
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English (en)
Finnish (fi)
Swedish (sv)
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FI950169A0 (fi
FI950169L (fi
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John L Krstenansky
Brian H Vickery
Jr John J Nestor
Teresa H Ho
Chinh T Bach
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Syntex Inc
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Publication of FI950169L publication Critical patent/FI950169L/fi
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Publication of FI120586B publication Critical patent/FI120586B/fi

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/635Parathyroid hormone, i.e. parathormone; Parathyroid hormone-related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/28Steroids, e.g. cholesterol, bile acids or glycyrrhetinic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40Cyclodextrins; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2319/00Fusion polypeptide

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Superconductors And Manufacturing Methods Therefor (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI950169A 1992-07-14 1995-01-13 Menetelmä PTH:n ja PTHRP:n analogien valmistamiseksi, ja niiden käyttö osteoporoosin hoitoon FI120586B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US07/915,247 US5589452A (en) 1992-07-14 1992-07-14 Analogs of parathyroid hormone and parathyroid hormone related peptide: synthesis and use for the treatment of osteoporosis
US91524792 1992-07-14
PCT/US1993/006465 WO1994001460A1 (en) 1992-07-14 1993-07-13 Analogs of pth and pthrp, their synthesis and use for the treatment of osteoporosis
US9306465 1993-07-13

Publications (3)

Publication Number Publication Date
FI950169A0 FI950169A0 (fi) 1995-01-13
FI950169L FI950169L (fi) 1995-01-13
FI120586B true FI120586B (fi) 2009-12-15

Family

ID=25435450

Family Applications (1)

Application Number Title Priority Date Filing Date
FI950169A FI120586B (fi) 1992-07-14 1995-01-13 Menetelmä PTH:n ja PTHRP:n analogien valmistamiseksi, ja niiden käyttö osteoporoosin hoitoon

Country Status (17)

Country Link
US (8) US5589452A (de)
EP (2) EP0651765B1 (de)
JP (1) JP4106082B2 (de)
KR (3) KR100458350B1 (de)
AT (1) ATE202115T1 (de)
AU (1) AU671851B2 (de)
CA (1) CA2140281C (de)
DE (1) DE69330347T2 (de)
DK (1) DK0651765T3 (de)
ES (1) ES2159293T3 (de)
FI (1) FI120586B (de)
GR (1) GR3036521T3 (de)
HU (2) HU217843B (de)
MX (1) MX9304226A (de)
NZ (1) NZ254554A (de)
PT (1) PT651765E (de)
WO (1) WO1994001460A1 (de)

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DK0651765T3 (da) 2001-09-24
US5589452A (en) 1996-12-31
US5807823A (en) 1998-09-15
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KR100404008B1 (ko) 2003-11-01
JP4106082B2 (ja) 2008-06-25
EP1094073A3 (de) 2002-09-25
EP1094073A2 (de) 2001-04-25
KR950702578A (ko) 1995-07-29
FI950169L (fi) 1995-01-13
DE69330347T2 (de) 2002-05-29
CA2140281A1 (en) 1994-01-20
NZ254554A (en) 1996-03-26
KR100458350B1 (ko) 2004-11-26
ATE202115T1 (de) 2001-06-15
US5693616A (en) 1997-12-02
US5840837A (en) 1998-11-24
HU217843B (hu) 2000-04-28
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MX9304226A (es) 1995-01-31
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HUT69628A (en) 1995-09-28
PT651765E (pt) 2001-11-30
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