JPS62277322A - 安定化された腸溶性抗潰瘍固形組成物 - Google Patents

安定化された腸溶性抗潰瘍固形組成物

Info

Publication number
JPS62277322A
JPS62277322A JP2999787A JP2999787A JPS62277322A JP S62277322 A JPS62277322 A JP S62277322A JP 2999787 A JP2999787 A JP 2999787A JP 2999787 A JP2999787 A JP 2999787A JP S62277322 A JPS62277322 A JP S62277322A
Authority
JP
Japan
Prior art keywords
compound
alkyl
magnesium
formula
examples
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2999787A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0338247B2 (fr
Inventor
Tadashi Makino
正 槙野
Tetsuro Tabata
哲朗 田畑
Shinichiro Hirai
真一郎 平井
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of JPS62277322A publication Critical patent/JPS62277322A/ja
Publication of JPH0338247B2 publication Critical patent/JPH0338247B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2999787A 1986-02-13 1987-02-12 安定化された腸溶性抗潰瘍固形組成物 Granted JPS62277322A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2956786 1986-02-13
JP61-29567 1986-02-13
JP61-38059 1986-02-21

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2316379A Division JPH0825905B2 (ja) 1990-11-20 1990-11-20 医薬固形組成物用安定化剤および安定化方法

Publications (2)

Publication Number Publication Date
JPS62277322A true JPS62277322A (ja) 1987-12-02
JPH0338247B2 JPH0338247B2 (fr) 1991-06-10

Family

ID=12279703

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2999787A Granted JPS62277322A (ja) 1986-02-13 1987-02-12 安定化された腸溶性抗潰瘍固形組成物

Country Status (1)

Country Link
JP (1) JPS62277322A (fr)

Cited By (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62258320A (ja) * 1986-04-30 1987-11-10 Yoshitomi Pharmaceut Ind Ltd 内服用新規医薬製剤
JPS62258316A (ja) * 1986-04-30 1987-11-10 Yoshitomi Pharmaceut Ind Ltd 酸不安定物質の内服用新規医薬製剤
JPH0222225A (ja) * 1988-07-11 1990-01-25 Eisai Co Ltd 胃酸分泌抑制剤含有固型製剤
JPH02138213A (ja) * 1988-08-18 1990-05-28 Takeda Chem Ind Ltd 注射剤
JPH03163018A (ja) * 1990-11-20 1991-07-15 Takeda Chem Ind Ltd 医薬固形組成物用安定化剤および安定化方法
JP2002114779A (ja) * 2000-08-04 2002-04-16 Takeda Chem Ind Ltd ベンズイミダゾール化合物の塩およびその用途
JP2004155773A (ja) * 2002-10-16 2004-06-03 Takeda Chem Ind Ltd 安定な固形製剤
US6780882B2 (en) 1996-01-04 2004-08-24 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
JP2006514049A (ja) * 2002-12-20 2006-04-27 タツプ・フアーマシユーテイカル・プロダクツ・インコーポレイテツド プロトンポンプ阻害剤、nsaid及び緩衝剤を含む剤形
JP2006515353A (ja) * 2003-01-15 2006-05-25 シプラ・リミテッド 製薬的方法、及び該方法により製造された化合物
JP2006528181A (ja) * 2003-07-18 2006-12-14 サンタラス インコーポレイティッド 酸分泌を阻害するために有用な薬学的製剤ならびにそれらを作製および使用する方法
EP1736144A2 (fr) 1998-05-18 2006-12-27 Takeda Pharmaceutical Company Limited Comprimé à désintégration orale
US7220762B1 (en) 1999-10-20 2007-05-22 Eisai R&D Management Co., Ltd. Methods for stabilizing benzimidazole compounds
WO2007074909A1 (fr) 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Preparation solide a liberation controlee
WO2007074856A1 (fr) 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Procede de production de preparation solide se desintegrant dans la cavite orale
WO2007074910A1 (fr) * 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Preparation solide a liberation controlee
JP2008530175A (ja) * 2005-02-16 2008-08-07 ソルヴェイ(ソシエテ アノニム) 生物学的活性物質と、炭酸カルシウム含有賦形剤とを含む錠剤
WO2008111278A1 (fr) * 2007-03-12 2008-09-18 Tomita Pharmaceutical Co., Ltd. Vecteur pharmaceutique et produit pharmaceutique
JP2008255088A (ja) * 2007-03-12 2008-10-23 Tomita Pharmaceutical Co Ltd 製剤用球形核粒子
WO2009069280A1 (fr) * 2007-11-27 2009-06-04 Ohara Pharmaceutical Co., Ltd. Procédé de production d'une substance granulée
JP2010180225A (ja) * 2002-10-16 2010-08-19 Takeda Chem Ind Ltd 安定な固形製剤
EP2258351A2 (fr) 2001-10-17 2010-12-08 Takeda Pharmaceutical Company Limited Granules contenant lansoprazol en grande quantité
EP2277510A2 (fr) 2002-10-16 2011-01-26 Takeda Pharmaceutical Company Limited Préparation à libération contrôlée.
US8124780B2 (en) 2005-04-15 2012-02-28 Eisai R&D Management Co., Ltd. Benzimidazole compound
WO2012091153A2 (fr) 2010-12-27 2012-07-05 Takeda Pharmaceutical Company Limited Comprimé orodispersible
USRE45198E1 (en) 1996-01-04 2014-10-14 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US9040564B2 (en) 2005-04-28 2015-05-26 Eisai R&D Management Co., Ltd. Stabilized composition
US9241910B2 (en) 2008-03-11 2016-01-26 Takeda Pharmaceutical Company Limited Orally-disintegrating solid preparation
WO2018229744A1 (fr) 2017-06-12 2018-12-20 Glytech Llc. Traitement de la dépression avec des antagonistes du nmda et de la d2/5ht2a ou des antagonistes de la 5ht2a sélectifs

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58135881A (ja) * 1981-11-05 1983-08-12 ビク−グルデン・ロムベルク・ヘミツシエ・フアブリク・ゲゼルシヤフト・ミト・ベシユレンクテル・ハフツング 置換ベンズイミダゾ−ル類、その製造方法と利用、およびこれを含む医薬
JPS59167587A (ja) * 1983-03-04 1984-09-21 アクチエボラゲツト・ヘツスレ オメプラゾ−ル化合物

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58135881A (ja) * 1981-11-05 1983-08-12 ビク−グルデン・ロムベルク・ヘミツシエ・フアブリク・ゲゼルシヤフト・ミト・ベシユレンクテル・ハフツング 置換ベンズイミダゾ−ル類、その製造方法と利用、およびこれを含む医薬
JPS59167587A (ja) * 1983-03-04 1984-09-21 アクチエボラゲツト・ヘツスレ オメプラゾ−ル化合物

Cited By (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62258316A (ja) * 1986-04-30 1987-11-10 Yoshitomi Pharmaceut Ind Ltd 酸不安定物質の内服用新規医薬製剤
JPS62258320A (ja) * 1986-04-30 1987-11-10 Yoshitomi Pharmaceut Ind Ltd 内服用新規医薬製剤
JPH0222225A (ja) * 1988-07-11 1990-01-25 Eisai Co Ltd 胃酸分泌抑制剤含有固型製剤
JPH02138213A (ja) * 1988-08-18 1990-05-28 Takeda Chem Ind Ltd 注射剤
JPH03163018A (ja) * 1990-11-20 1991-07-15 Takeda Chem Ind Ltd 医薬固形組成物用安定化剤および安定化方法
USRE45198E1 (en) 1996-01-04 2014-10-14 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US6780882B2 (en) 1996-01-04 2004-08-24 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
EP2263660A2 (fr) 1998-05-18 2010-12-22 Takeda Pharmaceutical Company Limited Comprimé se désintégrant dans la bouche
EP1736144A2 (fr) 1998-05-18 2006-12-27 Takeda Pharmaceutical Company Limited Comprimé à désintégration orale
US7220762B1 (en) 1999-10-20 2007-05-22 Eisai R&D Management Co., Ltd. Methods for stabilizing benzimidazole compounds
JP2002114779A (ja) * 2000-08-04 2002-04-16 Takeda Chem Ind Ltd ベンズイミダゾール化合物の塩およびその用途
EP2258351A2 (fr) 2001-10-17 2010-12-08 Takeda Pharmaceutical Company Limited Granules contenant lansoprazol en grande quantité
JP2010180225A (ja) * 2002-10-16 2010-08-19 Takeda Chem Ind Ltd 安定な固形製剤
EP2596792A1 (fr) 2002-10-16 2013-05-29 Takeda Pharmaceutical Company Limited Préparations solides stables
JP2004155773A (ja) * 2002-10-16 2004-06-03 Takeda Chem Ind Ltd 安定な固形製剤
US8697094B2 (en) 2002-10-16 2014-04-15 Takeda Pharmaceutical Company Limited Stable solid preparations
US8697097B2 (en) 2002-10-16 2014-04-15 Takeda Pharmaceutical Company Limited Stable solid preparations
JP2013151525A (ja) * 2002-10-16 2013-08-08 Takeda Chem Ind Ltd 安定な固形製剤
EP2596791A1 (fr) 2002-10-16 2013-05-29 Takeda Pharmaceutical Company Limited Préparations solides stables
JP2015145405A (ja) * 2002-10-16 2015-08-13 武田薬品工業株式会社 安定な固形製剤
US9265730B2 (en) 2002-10-16 2016-02-23 Takeda Pharmaceutical Company Limited Stable solid preparations
EP2283827A1 (fr) 2002-10-16 2011-02-16 Takeda Pharmaceutical Company Limited Préparation à libération contrôlée
EP2277510A2 (fr) 2002-10-16 2011-01-26 Takeda Pharmaceutical Company Limited Préparation à libération contrôlée.
JP2006514049A (ja) * 2002-12-20 2006-04-27 タツプ・フアーマシユーテイカル・プロダクツ・インコーポレイテツド プロトンポンプ阻害剤、nsaid及び緩衝剤を含む剤形
JP2012107021A (ja) * 2002-12-20 2012-06-07 Takeda Pharmaceuticals Usa Inc プロトンポンプ阻害剤、nsaid及び緩衝剤を含む剤形
JP2006515353A (ja) * 2003-01-15 2006-05-25 シプラ・リミテッド 製薬的方法、及び該方法により製造された化合物
JP2006528181A (ja) * 2003-07-18 2006-12-14 サンタラス インコーポレイティッド 酸分泌を阻害するために有用な薬学的製剤ならびにそれらを作製および使用する方法
US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
JP2008530175A (ja) * 2005-02-16 2008-08-07 ソルヴェイ(ソシエテ アノニム) 生物学的活性物質と、炭酸カルシウム含有賦形剤とを含む錠剤
US8124780B2 (en) 2005-04-15 2012-02-28 Eisai R&D Management Co., Ltd. Benzimidazole compound
US9040564B2 (en) 2005-04-28 2015-05-26 Eisai R&D Management Co., Ltd. Stabilized composition
WO2007074909A1 (fr) 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Preparation solide a liberation controlee
WO2007074910A1 (fr) * 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Preparation solide a liberation controlee
WO2007074856A1 (fr) 2005-12-28 2007-07-05 Takeda Pharmaceutical Company Limited Procede de production de preparation solide se desintegrant dans la cavite orale
JPWO2007074910A1 (ja) * 2005-12-28 2009-06-04 武田薬品工業株式会社 放出制御固形製剤
JPWO2007074909A1 (ja) * 2005-12-28 2009-06-04 武田薬品工業株式会社 放出制御固形製剤
WO2008111278A1 (fr) * 2007-03-12 2008-09-18 Tomita Pharmaceutical Co., Ltd. Vecteur pharmaceutique et produit pharmaceutique
JP2008255088A (ja) * 2007-03-12 2008-10-23 Tomita Pharmaceutical Co Ltd 製剤用球形核粒子
WO2009069280A1 (fr) * 2007-11-27 2009-06-04 Ohara Pharmaceutical Co., Ltd. Procédé de production d'une substance granulée
JPWO2009069280A1 (ja) * 2007-11-27 2011-04-07 大原薬品工業株式会社 造粒物の製造法
US9241910B2 (en) 2008-03-11 2016-01-26 Takeda Pharmaceutical Company Limited Orally-disintegrating solid preparation
WO2012091153A2 (fr) 2010-12-27 2012-07-05 Takeda Pharmaceutical Company Limited Comprimé orodispersible
WO2018229744A1 (fr) 2017-06-12 2018-12-20 Glytech Llc. Traitement de la dépression avec des antagonistes du nmda et de la d2/5ht2a ou des antagonistes de la 5ht2a sélectifs

Also Published As

Publication number Publication date
JPH0338247B2 (fr) 1991-06-10

Similar Documents

Publication Publication Date Title
JPS62277322A (ja) 安定化された腸溶性抗潰瘍固形組成物
DE3780045T2 (de) Verwendung von basischen anorganischen magnesium- oder calciumsalzen zur stabilisierung von benzimidazolderivaten.
US5879708A (en) Stabilized pharmaceutical composition
US6749864B2 (en) Stabilized pharmaceutical composition
HK1002021B (en) Stabilized pharmaceutical composition and its production
JP4834553B2 (ja) 医薬組成物
KR930010495B1 (ko) 피리딘 유도체의 제조방법
DE3530046C2 (de) Äthylendiaminmonoamid-Derivate
JP2762998B2 (ja) 医薬固形組成物用安定化剤および安定化方法
JPH03163018A (ja) 医薬固形組成物用安定化剤および安定化方法
JPS63502658A (ja) 新規な物質の組成
JPH10273440A (ja) ピリダジノン化合物類の経口製剤
CA1338377C (fr) Composition pharmaceutique stabilisee et sa preparation
KR950007211B1 (ko) 안전화된 약제 조성물 및 항궤양 약제 조성물의 안정화 방법
IE904248A1 (en) Therapeutically active fluoro substituted benzimidazoles,¹processes for their preparation as well as their use
JPH05112559A (ja) 4−アミノ−5−ピリミジンカルボン酸誘導体
JPH08311041A (ja) 複素環化合物およびその剤
JPH072636B2 (ja) 胃腸の細胞保護剤

Legal Events

Date Code Title Description
EXPY Cancellation because of completion of term