NO20051689L - Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister - Google Patents

Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister

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Publication number
NO20051689L
NO20051689L NO20051689A NO20051689A NO20051689L NO 20051689 L NO20051689 L NO 20051689L NO 20051689 A NO20051689 A NO 20051689A NO 20051689 A NO20051689 A NO 20051689A NO 20051689 L NO20051689 L NO 20051689L
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NO
Norway
Prior art keywords
histamine
antagonists
diaszepines
heptanes
diazabicyclo
Prior art date
Application number
NO20051689A
Other languages
English (en)
Other versions
NO20051689D0 (no
Inventor
Heather Hobbs
David Matthew Wilson
Rachael Anne Ancliff
Colin David Eldred
Simon Tennby Hodgson
Thomas Daniel Heightman
Yvonne C Fogden
Ashley Paul Hancock
Matthew J Lindon
Original Assignee
Glaxo Group Ltd
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Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20051689D0 publication Critical patent/NO20051689D0/no
Publication of NO20051689L publication Critical patent/NO20051689L/no

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Abstract

Foreliggende oppfinnelse vedrører nye piperazin- og azepinderivater med farmakologisk aktivitet, fremgangsmåter for fremstilling derav, sammensetninger som inneholder disse og anvendelse derav for behandling av nevrodegenerativeforstyrrelser inkludert Alzheimers sykdom.
NO20051689A 2002-10-16 2005-04-05 Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister NO20051689L (no)

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GBGB0224084.4A GB0224084D0 (en) 2002-10-16 2002-10-16 Novel compounds
PCT/EP2003/011423 WO2004035556A1 (en) 2002-10-16 2003-10-14 Substituted piperazines, (1,4) diaszepines, and 2,5-diazabicyclo (2.2.1) heptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists

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JP2006508935A (ja) 2006-03-16
NZ539446A (en) 2006-11-30
NO20051689D0 (no) 2005-04-05
CN100400523C (zh) 2008-07-09
ZA200603604B (en) 2007-04-25
JP2007016041A (ja) 2007-01-25
RU2005110061A (ru) 2006-01-20
CA2502249A1 (en) 2004-04-29
CN101070309A (zh) 2007-11-14
US20060025404A1 (en) 2006-02-02
IS7782A (is) 2005-03-31
EP1567511A1 (en) 2005-08-31
BR0315283A (pt) 2005-08-30
PL376477A1 (en) 2005-12-27
NZ549963A (en) 2008-03-28
RU2328494C2 (ru) 2008-07-10
CN1726201A (zh) 2006-01-25
KR20050049553A (ko) 2005-05-25
US7615550B2 (en) 2009-11-10
ZA200502873B (en) 2006-07-26
WO2004035556A1 (en) 2004-04-29
US20100075953A1 (en) 2010-03-25
AU2003280380A1 (en) 2004-05-04

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