OA10843A - Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma - Google Patents
Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma Download PDFInfo
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- OA10843A OA10843A OA9800148A OA9800148A OA10843A OA 10843 A OA10843 A OA 10843A OA 9800148 A OA9800148 A OA 9800148A OA 9800148 A OA9800148 A OA 9800148A OA 10843 A OA10843 A OA 10843A
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- OA
- OAPI
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- phenyl
- methyl
- ethoxy
- propionic acid
- phenylamino
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| EP0925063A4 (en) * | 1996-07-01 | 2000-12-27 | Lilly Co Eli | Blood-glucose-lowering and lipid-lowering compounds |
| EE03765B1 (et) * | 1996-08-19 | 2002-06-17 | Japan Tobacco Inc. | Propioonhappe derivaadid ja nende kasutamine |
| JP2001514663A (ja) | 1997-03-12 | 2001-09-11 | エスモンド,ロバート ダブリュー. | アルツハイマー病を処置または予防するための方法 |
| DE69815008T2 (de) * | 1997-09-19 | 2004-04-01 | Ssp Co., Ltd. | Alfa-substituierte Phenylpropionsäurederivate und diese enthaltende Arzneimittel |
| WO1999018066A1 (en) * | 1997-10-02 | 1999-04-15 | Sankyo Company, Limited | Amidocarboxylic acid derivatives |
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| US6329372B1 (en) * | 1998-01-27 | 2001-12-11 | Celltech Therapeutics Limited | Phenylalanine derivatives |
| EP1053227B1 (en) * | 1998-01-29 | 2008-11-05 | Amgen Inc. | Ppar-gamma modulators |
| US6583157B2 (en) | 1998-01-29 | 2003-06-24 | Tularik Inc. | Quinolinyl and benzothiazolyl modulators |
| ES2226413T3 (es) | 1998-02-26 | 2005-03-16 | Celltech Therapeutics Limited | Derivados de fenilalanina como inhibidores de alfa-4 integrinas. |
| GB9805655D0 (en) | 1998-03-16 | 1998-05-13 | Celltech Therapeutics Ltd | Chemical compounds |
| US6521626B1 (en) | 1998-03-24 | 2003-02-18 | Celltech R&D Limited | Thiocarboxamide derivatives |
| EP1077957B1 (en) * | 1998-05-11 | 2004-08-04 | Takeda Chemical Industries, Ltd. | Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity |
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| MA26634A1 (fr) * | 1998-06-04 | 2004-12-20 | Astra Ab | Nouveaux derives de l'acide 3-aryl propionique et analogues |
| RU2243214C2 (ru) * | 1998-06-04 | 2004-12-27 | Астразенека Аб | Новые производные и аналоги 3-арилпропионовой кислоты |
| SE9801992D0 (sv) | 1998-06-04 | 1998-06-04 | Astra Ab | New 3-aryl-2-hydroxypropionic acid derivative I |
| US7045519B2 (en) | 1998-06-19 | 2006-05-16 | Chiron Corporation | Inhibitors of glycogen synthase kinase 3 |
| CN1312807A (zh) * | 1998-06-19 | 2001-09-12 | 希龙公司 | 糖元合成酶激酶3的抑制剂 |
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| US6589969B1 (en) * | 1998-10-16 | 2003-07-08 | Ono Pharmaceutical Co., Ltd. | Carboxylic acid derivatives and drugs containing the same as the active ingredient |
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| JP2002532416A (ja) * | 1998-12-17 | 2002-10-02 | マインドセット・バイオファーマシューティカルズ・(ユーエスエイ)・インコーポレイテッド | 脳のグルコース利用の増進 |
| US6127394A (en) * | 1999-03-08 | 2000-10-03 | The University Of Mississippi | 1,2-Dithiolane derivatives |
| US6204288B1 (en) | 1999-03-08 | 2001-03-20 | The University Of Mississippi | 1,2-dithiolane derivatives |
| KR20020060067A (ko) * | 1999-04-06 | 2002-07-16 | 가와무라 요시부미 | α-치환 카르복실산 유도체 |
| HRP20010748A2 (en) * | 1999-04-16 | 2003-02-28 | Reddys Lab Ltd Dr | Novel polymorphic forms of an antidiabetic agent: process for their preparation and pharmaceutical compositions containing them |
| WO2000063189A1 (en) * | 1999-04-16 | 2000-10-26 | Novo Nordisk A/S | Crystalline r- guanidines, arginine or (l) -arginine (2s) -2- ethoxy -3-{4- [2-(10h -phenoxazin -10-yl)ethoxy]phenyl}propanoate |
| US6528507B1 (en) | 1999-04-16 | 2003-03-04 | Dr. Reddy's Laboratories Limited | Polymorphic forms of an antidiabetic agent: process for their preparation and a pharmaceutical composition containing them |
| CA2370742A1 (en) * | 1999-04-19 | 2000-10-26 | Coelacanth Corporation | Ppar-(gamma) agonists as agents for the treatment of type ii diabetes |
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| CN1348439A (zh) * | 1999-04-20 | 2002-05-08 | 诺沃挪第克公司 | 新化合物及其制备和用途 |
| US7414128B2 (en) | 1999-04-20 | 2008-08-19 | Dr. Reddy's Laboratories, Limited | Crystalline R-guanidines, Arginine or (L)-Arginine (2S)-2-Ethoxy-3-{4-[2-(10H -phenoxazin-10-yl)ethoxy]phenyl}propanoate |
| EP1171431A1 (en) * | 1999-04-20 | 2002-01-16 | Novo Nordisk A/S | Compounds, their preparation and use |
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| WO2000064876A1 (en) | 1999-04-28 | 2000-11-02 | Aventis Pharma Deutschland Gmbh | Tri-aryl acid derivatives as ppar receptor ligands |
| EP1175412A1 (en) * | 1999-04-28 | 2002-01-30 | Dr. Reddy's Research Foundation | Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents |
| US6518283B1 (en) | 1999-05-28 | 2003-02-11 | Celltech R&D Limited | Squaric acid derivatives |
| JP4618845B2 (ja) * | 1999-06-09 | 2011-01-26 | 杏林製薬株式会社 | ヒトペルオキシゾーム増殖薬活性化受容体(PPAR)αアゴニストとしての置換フェニルプロピオン酸誘導体 |
| GB9913782D0 (en) * | 1999-06-14 | 1999-08-11 | Smithkline Beecham Plc | Novel compounds |
| GB9914977D0 (en) * | 1999-06-25 | 1999-08-25 | Glaxo Group Ltd | Chemical compounds |
| CN1171872C (zh) * | 1999-06-30 | 2004-10-20 | 图拉列克股份有限公司 | 调节PPARγ活性的化合物 |
| US7041691B1 (en) | 1999-06-30 | 2006-05-09 | Amgen Inc. | Compounds for the modulation of PPARγ activity |
| AU7073400A (en) * | 1999-08-27 | 2001-03-26 | Eli Lilly And Company | Biaryl-oxa(thia)zole derivatives and their use as ppars modulators |
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- 1997-02-26 IL IL12579697A patent/IL125796A/en not_active IP Right Cessation
- 1997-02-26 US US09/125,750 patent/US6294580B1/en not_active Expired - Fee Related
- 1997-02-26 DE DE69706658T patent/DE69706658T2/de not_active Expired - Lifetime
- 1997-02-26 UA UA98084544A patent/UA58502C2/uk unknown
- 1997-02-26 BR BRPI9707786-0A patent/BR9707786B1/pt not_active IP Right Cessation
- 1997-02-26 EP EP97906130A patent/EP0888317B1/en not_active Expired - Lifetime
- 1997-02-26 SI SI9730233T patent/SI0888317T1/xx unknown
- 1997-02-26 PT PT97906130T patent/PT888317E/pt unknown
- 1997-02-26 CN CN97193988A patent/CN1093124C/zh not_active Expired - Fee Related
- 1997-02-26 PL PL328871A patent/PL191118B1/pl not_active IP Right Cessation
- 1997-02-26 TR TR1998/01707T patent/TR199801707T2/xx unknown
- 1997-02-26 WO PCT/EP1997/000916 patent/WO1997031907A1/en not_active Ceased
- 1997-02-27 ID IDP970584A patent/ID15985A/id unknown
- 1997-02-27 AR ARP970100771A patent/AR011502A1/es active IP Right Grant
- 1997-02-27 AP APAP/P/1997/000935A patent/AP780A/en active
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1998
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- 1998-08-25 OA OA9800148A patent/OA10843A/en unknown
- 1998-08-27 NO NO19983940A patent/NO311516B1/no not_active IP Right Cessation
- 1998-08-28 RS YUP-369/98A patent/RS49586B/sr unknown
- 1998-09-24 BG BG102792A patent/BG102792A/bg unknown
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2003
- 2003-03-12 CY CY0300026A patent/CY2319B1/xx unknown
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