ATE121730T1 - N-aryl und n-heteroarylamide und harnstoffderivate als inhibitoren von acyl- coenzym a: cholesterol-acyl-transferase. - Google Patents

N-aryl und n-heteroarylamide und harnstoffderivate als inhibitoren von acyl- coenzym a: cholesterol-acyl-transferase.

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Publication number
ATE121730T1
ATE121730T1 AT90310009T AT90310009T ATE121730T1 AT E121730 T1 ATE121730 T1 AT E121730T1 AT 90310009 T AT90310009 T AT 90310009T AT 90310009 T AT90310009 T AT 90310009T AT E121730 T1 ATE121730 T1 AT E121730T1
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Austria
Prior art keywords
acyl
inhibitors
coenzyme
cholesterol
heteroarylamide
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AT90310009T
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English (en)
Inventor
Peter A Mccarthy
Frederick J Walker
Thien Truong
Ernest S Hamanaka
George Chang
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Pfizer
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Publication of ATE121730T1 publication Critical patent/ATE121730T1/de

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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AT90310009T 1989-09-15 1990-09-13 N-aryl und n-heteroarylamide und harnstoffderivate als inhibitoren von acyl- coenzym a: cholesterol-acyl-transferase. ATE121730T1 (de)

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AT94200437T ATE177082T1 (de) 1989-09-15 1990-09-13 N-heteroarylamidederivate als inhibitoren von acyl-coenzym a: cholesterol-acyl-transferase
AT90310009T ATE121730T1 (de) 1989-09-15 1990-09-13 N-aryl und n-heteroarylamide und harnstoffderivate als inhibitoren von acyl- coenzym a: cholesterol-acyl-transferase.

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PL291470A1 (en) 1992-07-13
AU652345B2 (en) 1994-08-25
NO904022D0 (no) 1990-09-14
CA2025301A1 (en) 1991-03-16
HUT70027A (en) 1995-09-28
JPH03120243A (ja) 1991-05-22
AU6255390A (en) 1991-04-18
PT95310A (pt) 1991-05-22
PL291471A1 (en) 1992-06-26
FI111362B (fi) 2003-07-15
HU9302945D0 (en) 1993-12-28
ES2071033T3 (es) 1995-06-16
KR910006233A (ko) 1991-04-27
DK0418071T3 (da) 1995-09-04
MX22406A (es) 1994-01-31
PL291472A1 (en) 1992-07-13
IL95610A0 (en) 1991-06-30
WO1991004027A1 (en) 1991-04-04
IL110324A0 (en) 1994-10-21
IL110321A0 (en) 1994-10-21
EP0418071A3 (en) 1992-03-25
DD298092A5 (de) 1992-02-06
NO904022L (no) 1991-03-18
EP0609960B1 (de) 1999-03-03
IE903336A1 (en) 1991-04-10
IE66324B1 (en) 1995-12-27
DE69018908D1 (de) 1995-06-01
ATE177082T1 (de) 1999-03-15
PL165357B1 (pl) 1994-12-30
EP0418071A2 (de) 1991-03-20
JPH0825974B2 (ja) 1996-03-13
CA2025301C (en) 2001-10-16
ZA907346B (en) 1992-05-27
IL95610A (en) 1994-12-29
EP0609960A1 (de) 1994-08-10
DE69032981T2 (de) 1999-07-08
GR3029826T3 (en) 1999-06-30
ES2127878T3 (es) 1999-05-01
DE69032981D1 (de) 1999-04-08
KR930011303B1 (ko) 1993-11-29
PT95310B (pt) 1997-06-30
NZ235323A (en) 1993-02-25
EG19358A (en) 1994-12-30
EP0418071B1 (de) 1995-04-26
CN1050183A (zh) 1991-03-27
PL165370B1 (pl) 1994-12-30
DK0609960T3 (da) 1999-09-27
FI904537A0 (fi) 1990-09-14
DE69018908T2 (de) 1995-08-24

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