EG19358A - Process for preparing of new n- aryl and n- heteroaryla-mide and urea derivatives as inhibitors of acyl coenzymes a: cholesterol acyl transferase ( A C A T ) - Google Patents

Process for preparing of new n- aryl and n- heteroaryla-mide and urea derivatives as inhibitors of acyl coenzymes a: cholesterol acyl transferase ( A C A T )

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Publication number
EG19358A
EG19358A EG54590A EG54590A EG19358A EG 19358 A EG19358 A EG 19358A EG 54590 A EG54590 A EG 54590A EG 54590 A EG54590 A EG 54590A EG 19358 A EG19358 A EG 19358A
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EG
Egypt
Prior art keywords
acyl
inhibitors
heteroaryla
mide
aryl
Prior art date
Application number
EG54590A
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English (en)
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Pfizer
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Publication date
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Publication of EG19358A publication Critical patent/EG19358A/xx

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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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EG54590A 1989-09-15 1990-09-13 Process for preparing of new n- aryl and n- heteroaryla-mide and urea derivatives as inhibitors of acyl coenzymes a: cholesterol acyl transferase ( A C A T ) EG19358A (en)

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PCT/US1989/004033 WO1991004027A1 (en) 1989-09-15 1989-09-15 New n-aryl and n-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat)

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DE (2) DE69032981T2 (de)
DK (2) DK0418071T3 (de)
EG (1) EG19358A (de)
ES (2) ES2071033T3 (de)
FI (1) FI111362B (de)
GR (1) GR3029826T3 (de)
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KR20210020866A (ko) 2018-06-12 2021-02-24 브이티브이 테라퓨틱스 엘엘씨 인슐린 또는 인슐린 유사체와 조합된 글루코키나제 활성제의 치료적 용도
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HUT70027A (en) 1995-09-28
ES2071033T3 (es) 1995-06-16
WO1991004027A1 (en) 1991-04-04
DE69018908T2 (de) 1995-08-24
HU9302945D0 (en) 1993-12-28
DE69032981T2 (de) 1999-07-08
PL165370B1 (pl) 1994-12-30
DD298092A5 (de) 1992-02-06
IE66324B1 (en) 1995-12-27
EP0609960B1 (de) 1999-03-03
CA2025301C (en) 2001-10-16
ATE121730T1 (de) 1995-05-15
AU652345B2 (en) 1994-08-25
NO904022L (no) 1991-03-18
KR930011303B1 (ko) 1993-11-29
NO904022D0 (no) 1990-09-14
ATE177082T1 (de) 1999-03-15
NZ235323A (en) 1993-02-25
PL165357B1 (pl) 1994-12-30
IL110321A0 (en) 1994-10-21
PT95310B (pt) 1997-06-30
ZA907346B (en) 1992-05-27
CA2025301A1 (en) 1991-03-16
DK0418071T3 (da) 1995-09-04
EP0418071A2 (de) 1991-03-20
MX22406A (es) 1994-01-31
IL95610A0 (en) 1991-06-30
AU6255390A (en) 1991-04-18
DE69018908D1 (de) 1995-06-01
EP0609960A1 (de) 1994-08-10
CN1050183A (zh) 1991-03-27
IE903336A1 (en) 1991-04-10
EP0418071A3 (en) 1992-03-25
JPH03120243A (ja) 1991-05-22
JPH0825974B2 (ja) 1996-03-13
IL110324A0 (en) 1994-10-21
GR3029826T3 (en) 1999-06-30
EP0418071B1 (de) 1995-04-26
ES2127878T3 (es) 1999-05-01
DE69032981D1 (de) 1999-04-08
FI111362B (fi) 2003-07-15
IL95610A (en) 1994-12-29
PL291470A1 (en) 1992-07-13
PT95310A (pt) 1991-05-22
KR910006233A (ko) 1991-04-27
DK0609960T3 (da) 1999-09-27
PL291471A1 (en) 1992-06-26
FI904537A0 (fi) 1990-09-14
PL291472A1 (en) 1992-07-13

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