ATE127471T1 - Polyen-makrolidderivate. - Google Patents

Polyen-makrolidderivate.

Info

Publication number
ATE127471T1
ATE127471T1 AT90121400T AT90121400T ATE127471T1 AT E127471 T1 ATE127471 T1 AT E127471T1 AT 90121400 T AT90121400 T AT 90121400T AT 90121400 T AT90121400 T AT 90121400T AT E127471 T1 ATE127471 T1 AT E127471T1
Authority
AT
Austria
Prior art keywords
amines
partricin
radicals
reacting
prepared
Prior art date
Application number
AT90121400T
Other languages
English (en)
Inventor
Tiberio Bruzzese
Franco Ottoni
Giuseppe Ghielmetti
Original Assignee
Prodotti Antibiotici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Prodotti Antibiotici Spa filed Critical Prodotti Antibiotici Spa
Application granted granted Critical
Publication of ATE127471T1 publication Critical patent/ATE127471T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/10—Preparation of carboxylic acid amides from compounds not provided for in groups C07C231/02 - C07C231/08
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Communicable Diseases (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Steroid Compounds (AREA)
AT90121400T 1989-11-16 1990-11-08 Polyen-makrolidderivate. ATE127471T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02239689A IT1237772B (it) 1989-11-16 1989-11-16 Derivati di macrolidi polienici.

Publications (1)

Publication Number Publication Date
ATE127471T1 true ATE127471T1 (de) 1995-09-15

Family

ID=11195729

Family Applications (1)

Application Number Title Priority Date Filing Date
AT90121400T ATE127471T1 (de) 1989-11-16 1990-11-08 Polyen-makrolidderivate.

Country Status (9)

Country Link
US (1) US5296597A (de)
EP (1) EP0434943B1 (de)
JP (1) JP3094065B2 (de)
KR (1) KR0185200B1 (de)
AT (1) ATE127471T1 (de)
DE (1) DE69022196T2 (de)
ES (1) ES2079417T3 (de)
IT (1) IT1237772B (de)
PT (1) PT95910B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1243404B (it) * 1990-12-03 1994-06-10 Prodotti Antibiotici Spa Derivati della partricina
IT1283149B1 (it) * 1996-07-12 1998-04-07 Prodotti Antibiotici Spa Complessi di n'-dimetilaminoacetilpartricina a dimetilaminoetilamide, o suoi sali, e colesterol 3-solfato
IT1294740B1 (it) * 1997-09-16 1999-04-12 Prospa Bv Derivati della partricina per il trattamento profilattico e/o curativo delle contaminazioni fungine di colture cellulari e di tessuti
US6121244A (en) * 1997-09-19 2000-09-19 Prospa B.V. Antitumoral method by administration of partricin derivatives
AU780724B2 (en) 2000-01-14 2005-04-14 Migenix Inc. Derivatives of polyene macrolides and preparation and use thereof
US6664241B2 (en) * 2000-05-31 2003-12-16 Micrologix Biotech Inc. Water-soluble amide derivatives of polyene macrolides and preparation and uses thereof
ITMI20032280A1 (it) * 2003-11-24 2005-05-25 Tiberio Bruzzese Formulazioni farmaceutiche contenenti derivati della partricina e loro uso orale per il trattamento di infezioni fungine e protozoarie localizzate
MX365184B (es) * 2010-12-21 2019-05-21 Centro De Investig Y De Estudios Avanzados Del I P N Nuevos compuestos analogos de la anfotericina y composiciones farmaceuticas que los contienen.
GB201409451D0 (en) * 2014-05-28 2014-07-09 Ipabc Ltd Antimicrobial preparations, methods for preparing the same and uses thereof to combat microorganisms

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1406774A (en) * 1973-02-15 1975-09-17 Prodotti Antibiotici Spa Esters of patricin and of partricin derivatives
PL122086B1 (en) * 1979-04-09 1982-06-30 Politechnika Gdanska Process for preparing amides of antibiotics from the group of polyene macrolides and their derivativesvykh makrolidov i ikh proizvodnykh
JP5728715B2 (ja) 2011-08-11 2015-06-03 オリオン機械株式会社 乳量計

Also Published As

Publication number Publication date
EP0434943A1 (de) 1991-07-03
IT8922396A1 (it) 1991-05-16
KR0185200B1 (ko) 1999-05-15
DE69022196D1 (de) 1995-10-12
KR910009638A (ko) 1991-06-28
PT95910A (pt) 1991-09-13
EP0434943B1 (de) 1995-09-06
DE69022196T2 (de) 1996-02-01
ES2079417T3 (es) 1996-01-16
PT95910B (pt) 1998-01-30
IT8922396A0 (it) 1989-11-16
IT1237772B (it) 1993-06-17
JPH03188096A (ja) 1991-08-16
JP3094065B2 (ja) 2000-10-03
US5296597A (en) 1994-03-22

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EEIH Change in the person of patent owner
EEIH Change in the person of patent owner
EELA Cancelled due to lapse of time