ATE541845T1 - 2,3-substituierte azaindolderivate zur behandlung von virusinfektionen - Google Patents

2,3-substituierte azaindolderivate zur behandlung von virusinfektionen

Info

Publication number
ATE541845T1
ATE541845T1 AT08795630T AT08795630T ATE541845T1 AT E541845 T1 ATE541845 T1 AT E541845T1 AT 08795630 T AT08795630 T AT 08795630T AT 08795630 T AT08795630 T AT 08795630T AT E541845 T1 ATE541845 T1 AT E541845T1
Authority
AT
Austria
Prior art keywords
treatment
virus infections
azaindole derivatives
substituted azaindole
substituted
Prior art date
Application number
AT08795630T
Other languages
English (en)
Inventor
Gopinadhan Anilkumar
Stuart Rosenblum
Srikanth Venkatraman
F Njoroge
Joseph Kozlowski
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of ATE541845T1 publication Critical patent/ATE541845T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AT08795630T 2007-08-29 2008-08-27 2,3-substituierte azaindolderivate zur behandlung von virusinfektionen ATE541845T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US96870707P 2007-08-29 2007-08-29
PCT/US2008/010149 WO2009032125A1 (en) 2007-08-29 2008-08-27 2,3-substituted azaindole derivatives for treating viral infections

Publications (1)

Publication Number Publication Date
ATE541845T1 true ATE541845T1 (de) 2012-02-15

Family

ID=40227567

Family Applications (1)

Application Number Title Priority Date Filing Date
AT08795630T ATE541845T1 (de) 2007-08-29 2008-08-27 2,3-substituierte azaindolderivate zur behandlung von virusinfektionen

Country Status (15)

Country Link
US (1) US8404845B2 (de)
EP (1) EP2195317B1 (de)
JP (2) JP5258889B2 (de)
KR (1) KR20100065167A (de)
CN (1) CN101842374A (de)
AR (1) AR068108A1 (de)
AT (1) ATE541845T1 (de)
AU (1) AU2008295485B2 (de)
CA (1) CA2697500A1 (de)
CL (1) CL2008002540A1 (de)
MX (1) MX2010002318A (de)
PE (1) PE20090994A1 (de)
TW (1) TW200911807A (de)
WO (1) WO2009032125A1 (de)
ZA (1) ZA201001392B (de)

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ATE541845T1 (de) 2007-08-29 2012-02-15 Schering Corp 2,3-substituierte azaindolderivate zur behandlung von virusinfektionen
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EP2697242B1 (de) 2011-04-13 2018-10-03 Merck Sharp & Dohme Corp. 2'-azido-substituierte nukleosidderivate und verfahren zu ihrer verwendung zur behandlung von virenerkrankungen
BR112013026345A2 (pt) 2011-04-13 2019-04-24 Merck Sharp & Dohe Corp. composto, composição farmacêutica, uso de um composto, e, método para tratar um paciente infectado com hcv
WO2013033901A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Heterocyclic-substituted benzofuran derivatives and methods of use thereof for the treatment of viral diseases
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Also Published As

Publication number Publication date
PE20090994A1 (es) 2009-08-03
JP2013064013A (ja) 2013-04-11
MX2010002318A (es) 2010-03-22
WO2009032125A1 (en) 2009-03-12
CA2697500A1 (en) 2009-03-12
AU2008295485A1 (en) 2009-03-12
CN101842374A (zh) 2010-09-22
AU2008295485B2 (en) 2013-09-05
EP2195317B1 (de) 2012-01-18
US20100239527A1 (en) 2010-09-23
JP5258889B2 (ja) 2013-08-07
JP2010537982A (ja) 2010-12-09
TW200911807A (en) 2009-03-16
US8404845B2 (en) 2013-03-26
EP2195317A1 (de) 2010-06-16
ZA201001392B (en) 2010-11-24
AR068108A1 (es) 2009-11-04
CL2008002540A1 (es) 2009-07-17
KR20100065167A (ko) 2010-06-15

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