ECSP11011222A - Règimen de dosificaciòn para un agonista de los receptores de s1p - Google Patents

Règimen de dosificaciòn para un agonista de los receptores de s1p

Info

Publication number
ECSP11011222A
ECSP11011222A EC2011011222A ECSP11011222A ECSP11011222A EC SP11011222 A ECSP11011222 A EC SP11011222A EC 2011011222 A EC2011011222 A EC 2011011222A EC SP11011222 A ECSP11011222 A EC SP11011222A EC SP11011222 A ECSP11011222 A EC SP11011222A
Authority
EC
Ecuador
Prior art keywords
dosage scheme
dosage
receiver agonist
agonist
receiver
Prior art date
Application number
EC2011011222A
Other languages
English (en)
Inventor
Robert Schmouder
Thomas Dumortier
Olivier David
Michael Looby
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41667217&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP11011222(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ECSP11011222A publication Critical patent/ECSP11011222A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/661Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/10Phosphatides, e.g. lecithin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Los modulares o agonistas de los receptores de S1P se administran siguiendo un règimen de dosificaciòn en donde, durante los dias iniciales del tratamiento, la dosificaciòn diaria es màs baja que la dosificaciòn diaria convencional.
EC2011011222A 2008-12-22 2011-06-22 Règimen de dosificaciòn para un agonista de los receptores de s1p ECSP11011222A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13967208P 2008-12-22 2008-12-22
US21853009P 2009-06-19 2009-06-19
US24671509P 2009-09-29 2009-09-29

Publications (1)

Publication Number Publication Date
ECSP11011222A true ECSP11011222A (es) 2011-08-31

Family

ID=41667217

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2011011222A ECSP11011222A (es) 2008-12-22 2011-06-22 Règimen de dosificaciòn para un agonista de los receptores de s1p

Country Status (43)

Country Link
US (12) US20110257133A1 (es)
EP (7) EP3120844A1 (es)
JP (7) JP2012513401A (es)
KR (1) KR101347919B1 (es)
CN (1) CN102264359A (es)
AR (1) AR074826A1 (es)
AU (1) AU2009330176C9 (es)
BR (1) BRPI0923500A2 (es)
CA (1) CA2747802C (es)
CL (2) CL2011001529A1 (es)
CO (1) CO6390117A2 (es)
CR (1) CR20110274A (es)
CU (1) CU20110136A7 (es)
CY (5) CY1116990T1 (es)
DK (4) DK3453387T3 (es)
EA (1) EA201100978A1 (es)
EC (1) ECSP11011222A (es)
ES (4) ES2810823T3 (es)
FI (2) FI4098256T3 (es)
FR (2) FR20C1060I1 (es)
HN (1) HN2011001759A (es)
HR (4) HRP20151190T1 (es)
HU (6) HUE048717T4 (es)
IL (3) IL213170A0 (es)
LT (5) LT3453387T (es)
LU (1) LUC00183I2 (es)
MA (1) MA32981B1 (es)
ME (2) ME03594B (es)
MX (3) MX2011006623A (es)
NO (1) NO2020038I1 (es)
NZ (1) NZ593065A (es)
PE (1) PE20120337A1 (es)
PL (4) PL3453387T3 (es)
PT (4) PT3453387T (es)
RS (3) RS66784B9 (es)
SG (1) SG171404A1 (es)
SI (4) SI2379067T1 (es)
SM (2) SMT202000441T1 (es)
TN (1) TN2011000272A1 (es)
TW (1) TW201028143A (es)
UY (1) UY32352A (es)
WO (1) WO2010075239A1 (es)
ZA (2) ZA201103863B (es)

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FR2968556B1 (fr) 2010-12-13 2013-12-27 Centre Nat Rech Scient Inhibiteurs des infections a vih et leurs utilisations
BR112013017302B1 (pt) 2011-01-07 2021-12-07 Novartis Ag Composição farmacêutica em fase sólida
JP6133790B2 (ja) 2011-02-18 2017-05-24 ザ スクリプス リサーチ インスティテュート ミエリン形成細胞運命へのオリゴデンドロサイト前駆細胞の定方向分化
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EP2964249A1 (en) * 2013-03-06 2016-01-13 Acorda Therapeutics, Inc. Therapeutic dosing of a neuregulin or a fragment thereof for treatment or prophylaxis of heart failure
JP6401257B2 (ja) 2013-10-11 2018-10-10 テイコク ファーマ ユーエスエー インコーポレーテッド 局所用スフィンゴシン−1−リン酸受容体アゴニスト製剤及びその使用方法
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MX2016013245A (es) * 2014-04-10 2017-01-16 Novartis Ag Regimen de dosificacion de liberacion inmediata de moduladores s1p.
EP4056179A1 (en) 2014-12-11 2022-09-14 Actelion Pharmaceuticals Ltd Dosing regimen for ponesimod, a selective s1p1 receptor agonist
MA41139B1 (fr) 2014-12-11 2026-02-27 Laboratoires Juvise Pharmaceuticals Combinaison pharmaceutique comprenant du ponesimod et son utilisation dans le traitement de la sclérose en plaque
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RS66784B9 (sr) 2008-12-22 2025-08-29 Novartis Ag Režim doziranјa agonista s1p receptora

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SMT202000054T1 (it) 2020-03-13
HRP20201167T1 (hr) 2020-12-11
CY1122812T1 (el) 2021-05-05
EP4098256B1 (en) 2025-02-26
HUE052048T2 (hu) 2021-04-28
EP2379067B1 (en) 2015-09-02
JP2017141238A (ja) 2017-08-17
LTPA2025520I1 (es) 2025-06-25
HN2011001759A (es) 2013-11-26
US20200330407A1 (en) 2020-10-22
FR25C1012I1 (fr) 2025-06-13
US20110257133A1 (en) 2011-10-20
LT3453387T (lt) 2020-08-25
JP2016135752A (ja) 2016-07-28
US20250262171A1 (en) 2025-08-21
CL2013001558A1 (es) 2013-10-25
EP3409274A1 (en) 2018-12-05
MX2011006623A (es) 2011-07-12
RS66784B9 (sr) 2025-08-29
JP2019167360A (ja) 2019-10-03
FIC20253002I1 (fi) 2025-05-23
PT3453387T (pt) 2020-08-11
ZA201205942B (en) 2013-03-27
SI4098256T1 (sl) 2025-06-30
EP3409274B1 (en) 2019-11-20
PE20120337A1 (es) 2012-04-24
ME03594B (me) 2020-07-20
DK3453387T3 (da) 2020-08-10
DK4098256T3 (da) 2025-04-22
TN2011000272A1 (en) 2012-12-17
AU2009330176A1 (en) 2011-07-07
EP4098256B9 (en) 2025-06-18
EA201100978A1 (ru) 2012-01-30
LTPA2020005I1 (lt) 2020-12-10
HRP20151190T1 (hr) 2016-01-01
RS59857B1 (sr) 2020-02-28
EP3453387A1 (en) 2019-03-13
JP2014144970A (ja) 2014-08-14
ES2552823T3 (es) 2015-12-02
US20140148415A1 (en) 2014-05-29
HUE048717T4 (hu) 2022-02-28
ES2760607T3 (es) 2020-05-14
SI3453387T1 (sl) 2020-10-30
FR20C1060I1 (fr) 2020-12-25
PL4098256T3 (pl) 2025-06-09
NO2020038I1 (no) 2020-11-18
PT3409274T (pt) 2019-12-17
EP4098256A1 (en) 2022-12-07
SG171404A1 (en) 2011-07-28
ZA201103863B (en) 2012-10-31
HUE071189T2 (hu) 2025-08-28
CR20110274A (es) 2011-07-19
JP7329965B2 (ja) 2023-08-21
DK2379067T3 (en) 2015-12-07
US20190091180A1 (en) 2019-03-28
CY1123255T1 (el) 2021-10-29
SI3409274T1 (sl) 2020-03-31
NZ593065A (en) 2012-11-30
TW201028143A (en) 2010-08-01
MA32981B1 (fr) 2012-01-02
LUC00183I2 (es) 2024-07-01
WO2010075239A1 (en) 2010-07-01
CA2747802C (en) 2021-02-09
PT4098256T (pt) 2025-04-10
US20180289638A1 (en) 2018-10-11
IL274756A (en) 2020-07-30
AU2009330176C9 (en) 2017-01-05
EP3120844A1 (en) 2017-01-25
CY2020036I1 (el) 2021-03-12
AU2009330176B2 (en) 2014-03-06
LT4098256T (lt) 2025-06-10
MX2021010759A (es) 2022-07-19
PL3453387T3 (pl) 2020-11-02
AR074826A1 (es) 2011-02-16
CU20110136A7 (es) 2012-01-31
RS60666B1 (sr) 2020-09-30
PL3409274T3 (pl) 2020-06-01
ES2810823T3 (es) 2021-03-09
MX385959B (es) 2025-03-18
US20100160259A1 (en) 2010-06-24
CO6390117A2 (es) 2012-02-29
JP2012513401A (ja) 2012-06-14
HUS2000046I1 (hu) 2020-12-28
US20160081949A1 (en) 2016-03-24
CY2025012I1 (el) 2026-02-25
KR20110096175A (ko) 2011-08-29
SMT202000441T1 (it) 2020-09-10
CA2747802A1 (en) 2010-07-01
EP2907511A1 (en) 2015-08-19
KR101347919B1 (ko) 2014-01-07
PL2379067T3 (pl) 2016-02-29
CY1116990T1 (el) 2017-04-05
US20140066657A1 (en) 2014-03-06
DK4098256T5 (da) 2025-07-21
CN102264359A (zh) 2011-11-30
HUE026869T2 (en) 2016-08-29
HRP20192175T1 (hr) 2020-03-20
US20170189353A1 (en) 2017-07-06
IL278914A (en) 2021-01-31
LT3409274T (lt) 2020-02-10
US20220142949A1 (en) 2022-05-12
FI4098256T3 (fi) 2025-03-31
CL2011001529A1 (es) 2012-02-24
EP3453387B1 (en) 2020-06-03
PT2379067E (pt) 2015-12-23
RS66784B1 (sr) 2025-06-30
CY2020036I2 (el) 2021-06-25
HRP20250568T1 (hr) 2025-07-04
AU2009330176C1 (en) 2016-12-08
US20160263061A1 (en) 2016-09-15
ES3017254T3 (en) 2025-05-12
JP2022103194A (ja) 2022-07-07
CY2025012I2 (el) 2026-02-25
HUE048717T2 (hu) 2020-08-28
ME03802B (me) 2021-04-20
HUS2500026I1 (hu) 2025-07-28
EP2379067A1 (en) 2011-10-26
IL213170A0 (en) 2011-07-31
SI2379067T1 (sl) 2016-01-29
DK3409274T3 (da) 2019-12-16
UY32352A (es) 2010-07-30
JP2024129030A (ja) 2024-09-26
BRPI0923500A2 (pt) 2018-05-29
EP3677260A1 (en) 2020-07-08

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