IL118045A - History 4-Anilinoquinazoline, their preparation and the pharmaceutical preparations that make them up - Google Patents

History 4-Anilinoquinazoline, their preparation and the pharmaceutical preparations that make them up

Info

Publication number
IL118045A
IL118045A IL11804596A IL11804596A IL118045A IL 118045 A IL118045 A IL 118045A IL 11804596 A IL11804596 A IL 11804596A IL 11804596 A IL11804596 A IL 11804596A IL 118045 A IL118045 A IL 118045A
Authority
IL
Israel
Prior art keywords
alkoxy
formula
chloro
pharmaceutically
quinazoline
Prior art date
Application number
IL11804596A
Other languages
English (en)
Hebrew (he)
Other versions
IL118045A0 (en
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10773597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL118045(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of IL118045A0 publication Critical patent/IL118045A0/xx
Publication of IL118045A publication Critical patent/IL118045A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL11804596A 1995-04-27 1996-04-26 History 4-Anilinoquinazoline, their preparation and the pharmaceutical preparations that make them up IL118045A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9508538.7A GB9508538D0 (en) 1995-04-27 1995-04-27 Quinazoline derivatives

Publications (2)

Publication Number Publication Date
IL118045A0 IL118045A0 (en) 1996-08-04
IL118045A true IL118045A (en) 2001-10-31

Family

ID=10773597

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11804596A IL118045A (en) 1995-04-27 1996-04-26 History 4-Anilinoquinazoline, their preparation and the pharmaceutical preparations that make them up

Country Status (38)

Country Link
US (1) US5770599A (pl)
EP (1) EP0823900B1 (pl)
JP (1) JP3040486B2 (pl)
KR (1) KR100296656B1 (pl)
CN (1) CN1100046C (pl)
AR (1) AR003944A1 (pl)
AT (1) ATE198329T1 (pl)
AU (1) AU699163B2 (pl)
BG (1) BG62730B1 (pl)
BR (1) BRPI9608082B8 (pl)
CA (1) CA2215732C (pl)
CZ (1) CZ288489B6 (pl)
DE (2) DE122009000076I1 (pl)
DK (1) DK0823900T3 (pl)
EE (1) EE03482B1 (pl)
EG (1) EG24134A (pl)
ES (1) ES2153098T3 (pl)
FR (1) FR09C0065I2 (pl)
GB (1) GB9508538D0 (pl)
GR (1) GR3035211T3 (pl)
HR (1) HRP960204B1 (pl)
HU (1) HU223313B1 (pl)
IL (1) IL118045A (pl)
LU (1) LU91631I2 (pl)
MY (1) MY114425A (pl)
NL (1) NL300429I1 (pl)
NO (2) NO309472B1 (pl)
NZ (1) NZ305444A (pl)
PL (1) PL189182B1 (pl)
PT (1) PT823900E (pl)
RO (1) RO117849B1 (pl)
RU (1) RU2153495C2 (pl)
SI (1) SI0823900T1 (pl)
SK (1) SK282236B6 (pl)
TW (1) TW436486B (pl)
UA (1) UA52602C2 (pl)
WO (1) WO1996033980A1 (pl)
ZA (1) ZA963358B (pl)

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FR09C0065I2 (fr) 2014-03-28
EP0823900B1 (en) 2000-12-27
LU91631I2 (fr) 2010-02-17
HK1005371A1 (en) 1999-01-08
DE69611361T2 (de) 2001-04-26
US5770599A (en) 1998-06-23
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CA2215732C (en) 2002-04-09
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BRPI9608082B8 (pt) 2021-07-06
KR100296656B1 (ko) 2001-08-07
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MY114425A (en) 2002-10-31
HRP960204A2 (en) 1997-08-31
UA52602C2 (uk) 2003-01-15
GB9508538D0 (en) 1995-06-14
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