MA26700A1 - FORMULATIONS PHARMACEUTIQUES D'INHIBITEURS DE PDE-5 DE GMPc à LIBERATION CONTROLEE, ET PROCEDE POUR LEUR PREPARATION. - Google Patents

FORMULATIONS PHARMACEUTIQUES D'INHIBITEURS DE PDE-5 DE GMPc à LIBERATION CONTROLEE, ET PROCEDE POUR LEUR PREPARATION.

Info

Publication number
MA26700A1
MA26700A1 MA25820A MA25820A MA26700A1 MA 26700 A1 MA26700 A1 MA 26700A1 MA 25820 A MA25820 A MA 25820A MA 25820 A MA25820 A MA 25820A MA 26700 A1 MA26700 A1 MA 26700A1
Authority
MA
Morocco
Prior art keywords
inhibitors
preparation
controlled release
pharmaceutical formulations
pde
Prior art date
Application number
MA25820A
Other languages
English (en)
Inventor
King Elizabeth
James Macrae Ross
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA26700(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of MA26700A1 publication Critical patent/MA26700A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

DEPOSANT Société dite : PFIZER RESEARCH AND DEVELOPMENT COMPANY, N.V./S.A. REVENDICATION DE PRIORITES GB 23/10/1998 9823192.1 GB 27/10/1998 9826392.4 GB 16/11/1998 9825117.6 Voir en annexe le titre de l'invention et le texte de l'abrégé Formulations pharmaceutiques d'inhibiteurs de PDE-5 de GMPc à libération contrôlée,et procédé pour leur préparation L'invention concerne des formulations à libération contrôlée contenant un inhibiteur de PDE-5 de GMPc, pour l'administration orale. Elle concerne également un procédé pour leur préparation. Application : utilisation de ces formulations dans le traitement ou la prévention d'un dysfonctionnement sexuel.
MA25820A 1998-10-23 1999-10-20 FORMULATIONS PHARMACEUTIQUES D'INHIBITEURS DE PDE-5 DE GMPc à LIBERATION CONTROLEE, ET PROCEDE POUR LEUR PREPARATION. MA26700A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
MA26700A1 true MA26700A1 (fr) 2004-12-20

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25820A MA26700A1 (fr) 1998-10-23 1999-10-20 FORMULATIONS PHARMACEUTIQUES D'INHIBITEURS DE PDE-5 DE GMPc à LIBERATION CONTROLEE, ET PROCEDE POUR LEUR PREPARATION.

Country Status (44)

Country Link
US (1) US6964780B1 (fr)
EP (1) EP1123088B1 (fr)
JP (1) JP2002528408A (fr)
KR (1) KR20010075659A (fr)
CN (1) CN1324233A (fr)
AP (1) AP2001002125A0 (fr)
AT (1) ATE340562T1 (fr)
AU (1) AU756509B2 (fr)
BG (1) BG65323B1 (fr)
BR (1) BR9914718A (fr)
CA (1) CA2348086C (fr)
CO (1) CO5160262A1 (fr)
CR (1) CR6326A (fr)
CY (1) CY1106239T1 (fr)
CZ (1) CZ20011427A3 (fr)
DE (1) DE69933383T2 (fr)
DK (1) DK1123088T3 (fr)
DZ (1) DZ2923A1 (fr)
EA (1) EA004068B1 (fr)
EE (1) EE200100235A (fr)
ES (1) ES2272082T3 (fr)
GT (1) GT199900184A (fr)
HK (1) HK1041818A1 (fr)
HR (1) HRP20010285A2 (fr)
HU (1) HUP0104318A3 (fr)
ID (1) ID28232A (fr)
IL (1) IL141764A (fr)
IS (1) IS5865A (fr)
MA (1) MA26700A1 (fr)
MX (1) MXPA01004011A (fr)
MY (1) MY130727A (fr)
NO (1) NO20011933L (fr)
NZ (1) NZ510275A (fr)
OA (1) OA11664A (fr)
PA (1) PA8484301A1 (fr)
PE (1) PE20001286A1 (fr)
PL (1) PL195789B1 (fr)
PT (1) PT1123088E (fr)
SK (1) SK286473B6 (fr)
TR (1) TR200101103T2 (fr)
TW (1) TW577756B (fr)
UA (1) UA67802C2 (fr)
UY (1) UY25765A1 (fr)
WO (1) WO2000024383A1 (fr)

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US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
ATE552013T1 (de) 2000-09-06 2012-04-15 Mitsubishi Tanabe Pharma Corp Zubereitungen zur oralen anwendung
EP2283829A1 (fr) 2000-10-30 2011-02-16 Euro-Celtique S.A. Formulations d'hydrocodone à liberation lente
EP1366760B1 (fr) * 2001-02-15 2010-06-30 Mitsubishi Tanabe Pharma Corporation Comprimes a dissolution rapide dans la cavite buccale
US10675280B2 (en) 2001-10-20 2020-06-09 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin
UA78974C2 (en) 2001-10-20 2007-05-10 Boehringer Ingelheim Pharma Use of flibanserin for treating disorders of sexual desire
ITMI20020515A1 (it) * 2002-03-12 2003-09-12 Jagotec Ag Sistema per il rilasco controllato di uno o piu' principi attivi
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NZ551356A (en) 2004-05-11 2009-09-25 Emotional Brain Bv Pharmaceutical formulations and uses thereof in the treatment of female sexual dysfunction
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EP1790343A1 (fr) * 2005-11-11 2007-05-30 Emotional Brain B.V. Compositions pharmaceutiques et leur utilisation pour le traitement des dysfonctions sexuelles chez la femme
WO2008000760A1 (fr) 2006-06-30 2008-01-03 Boehringer Ingelheim International Gmbh Flibansérine dans le traitement de l'incontinence urinaire et des maladies associées
BRPI0716439B8 (pt) 2006-08-14 2021-05-25 Boehringer Ingelheim Int sistemas de liberação farmacêutico compreendendo flibanserina, processo para preparação e uso dos mesmos
BRPI0716436B8 (pt) 2006-08-25 2021-05-25 Boehringer Ingelheim Int sistema de liberação controlada e método para fabricação do mesmo
EP1925307A1 (fr) * 2006-11-03 2008-05-28 Emotional Brain B.V. Utilisation de 3-alpha-androstanediol pour le traitement des dysfonctions sexuelles
US20080226715A1 (en) * 2007-03-16 2008-09-18 Albert Cha Therapeutic compositions and methods
EP2167057A1 (fr) * 2007-06-13 2010-03-31 Bayer HealthCare AG Inhibiteurs de la phosphodiestérase (pde) destinés au traitement des troubles de l'audition
CL2008002693A1 (es) 2007-09-12 2009-10-16 Boehringer Ingelheim Int Uso de flibanserina para el tratamiento de sintomas vasomotores seleccionados de sofocos, sudores nocturnos, cambios de estado de animo e irritabilidad
US20110033506A1 (en) * 2008-02-08 2011-02-10 Adel Penhasi Combination dosage form of low-dose modafinil and low-dose sildenafil
EP2374460A4 (fr) * 2008-12-12 2013-08-21 Rhein Siegfried Sa De Cv Composition de sildénafil à libération pulsée et son procédé de préparation
KR101004205B1 (ko) * 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EA015250B9 (ru) * 2010-11-19 2013-10-30 Тева Фармасьютикал Индастриз, Лтд. Таблетка силденафила, обеспечивающая модифицированную фармакокинетику, и способ ее изготовления
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Also Published As

Publication number Publication date
OA11664A (en) 2005-01-07
MXPA01004011A (es) 2003-03-10
UY25765A1 (es) 2001-08-27
IL141764A0 (en) 2002-03-10
HK1041818A1 (zh) 2002-07-26
CZ20011427A3 (cs) 2001-10-17
GT199900184A (es) 2001-04-14
DE69933383D1 (de) 2006-11-09
NO20011933L (no) 2001-06-25
TR200101103T2 (tr) 2001-09-21
CA2348086C (fr) 2007-01-23
EE200100235A (et) 2002-08-15
EA004068B1 (ru) 2003-12-25
CN1324233A (zh) 2001-11-28
EP1123088A1 (fr) 2001-08-16
CY1106239T1 (el) 2011-06-08
IS5865A (is) 2001-02-27
CR6326A (es) 2004-02-23
SK5192001A3 (en) 2002-09-10
ES2272082T3 (es) 2007-04-16
CA2348086A1 (fr) 2000-05-04
ATE340562T1 (de) 2006-10-15
AU5878799A (en) 2000-05-15
EP1123088B1 (fr) 2006-09-27
PE20001286A1 (es) 2000-11-22
NO20011933D0 (no) 2001-04-19
US6964780B1 (en) 2005-11-15
HRP20010285A2 (en) 2002-06-30
EA200100298A1 (ru) 2001-08-27
KR20010075659A (ko) 2001-08-09
ID28232A (id) 2001-05-10
HUP0104318A2 (hu) 2002-03-28
MY130727A (en) 2007-07-31
HUP0104318A3 (en) 2003-12-29
TW577756B (en) 2004-03-01
BR9914718A (pt) 2001-07-10
PL347476A1 (en) 2002-04-08
NZ510275A (en) 2003-07-25
BG105465A (bg) 2001-12-29
BG65323B1 (bg) 2008-02-29
DZ2923A1 (fr) 2004-03-01
UA67802C2 (uk) 2004-07-15
AU756509B2 (en) 2003-01-16
SK286473B6 (sk) 2008-11-06
IL141764A (en) 2008-06-05
JP2002528408A (ja) 2002-09-03
DK1123088T3 (da) 2007-01-02
DE69933383T2 (de) 2007-02-01
WO2000024383A1 (fr) 2000-05-04
PT1123088E (pt) 2007-01-31
CO5160262A1 (es) 2002-05-30
PA8484301A1 (es) 2000-09-29
PL195789B1 (pl) 2007-10-31
AP2001002125A0 (en) 2001-04-04

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