NO20091862L - N-(3-bensyl) -2, 2- (bis-fenyl) - propan-1-amin derivativer som CETP inhibitorer for behandlingen av atherosclerose and cardiovaskulaere sykdommer - Google Patents
N-(3-bensyl) -2, 2- (bis-fenyl) - propan-1-amin derivativer som CETP inhibitorer for behandlingen av atherosclerose and cardiovaskulaere sykdommerInfo
- Publication number
- NO20091862L NO20091862L NO20091862A NO20091862A NO20091862L NO 20091862 L NO20091862 L NO 20091862L NO 20091862 A NO20091862 A NO 20091862A NO 20091862 A NO20091862 A NO 20091862A NO 20091862 L NO20091862 L NO 20091862L
- Authority
- NO
- Norway
- Prior art keywords
- propan
- atherosclerosis
- benzyl
- bis
- phenyl
- Prior art date
Links
- 201000001320 Atherosclerosis Diseases 0.000 title 1
- 208000024172 Cardiovascular disease Diseases 0.000 title 1
- 239000003354 cholesterol ester transfer protein inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
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- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
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- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
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- C07D239/32—One oxygen, sulfur or nitrogen atom
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- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
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- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/26—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D307/30—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/32—Oxygen atoms
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- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D309/04—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D309/14—Nitrogen atoms not forming part of a nitro radical
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- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
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- C07C2601/00—Systems containing only non-condensed rings
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- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
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- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86811206P | 2006-12-01 | 2006-12-01 | |
| PCT/US2007/085733 WO2008070496A2 (en) | 2006-12-01 | 2007-11-28 | N- ( (3-benzyl) -2, 2- (bis-phenyl) -propan-1-amine derivatives as cetp inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20091862L true NO20091862L (no) | 2009-08-19 |
Family
ID=39365913
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20091862A NO20091862L (no) | 2006-12-01 | 2009-05-13 | N-(3-bensyl) -2, 2- (bis-fenyl) - propan-1-amin derivativer som CETP inhibitorer for behandlingen av atherosclerose and cardiovaskulaere sykdommer |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US8404896B2 (de) |
| EP (1) | EP2094643B1 (de) |
| JP (2) | JP5498168B2 (de) |
| CN (1) | CN101663262B (de) |
| AT (1) | ATE547394T1 (de) |
| ES (1) | ES2382009T3 (de) |
| NO (1) | NO20091862L (de) |
| WO (1) | WO2008070496A2 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE547394T1 (de) * | 2006-12-01 | 2012-03-15 | Bristol Myers Squibb Co | N-((3-benzyl)-2,2-(bis-phenyl)-propan-1- aminderivate als cetp-hemmer für die behandlung von atherosklerose und herz-kreislauf- erkrankungen |
| EP2582709B1 (de) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
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-
2007
- 2007-11-28 AT AT07864837T patent/ATE547394T1/de active
- 2007-11-28 WO PCT/US2007/085733 patent/WO2008070496A2/en not_active Ceased
- 2007-11-28 ES ES07864837T patent/ES2382009T3/es active Active
- 2007-11-28 CN CN200780050689.7A patent/CN101663262B/zh not_active Expired - Fee Related
- 2007-11-28 EP EP07864837A patent/EP2094643B1/de active Active
- 2007-11-28 US US12/516,586 patent/US8404896B2/en active Active
- 2007-11-28 JP JP2009539455A patent/JP5498168B2/ja not_active Expired - Fee Related
-
2009
- 2009-05-13 NO NO20091862A patent/NO20091862L/no not_active Application Discontinuation
-
2012
- 2012-12-18 US US13/717,871 patent/US9102599B2/en active Active
-
2014
- 2014-01-28 JP JP2014013469A patent/JP2014098008A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US9102599B2 (en) | 2015-08-11 |
| WO2008070496A3 (en) | 2008-09-18 |
| EP2094643A2 (de) | 2009-09-02 |
| ES2382009T3 (es) | 2012-06-04 |
| CN101663262B (zh) | 2014-03-26 |
| US8404896B2 (en) | 2013-03-26 |
| US20130184279A1 (en) | 2013-07-18 |
| JP5498168B2 (ja) | 2014-05-21 |
| EP2094643B1 (de) | 2012-02-29 |
| JP2010511624A (ja) | 2010-04-15 |
| US20100041717A1 (en) | 2010-02-18 |
| CN101663262A (zh) | 2010-03-03 |
| WO2008070496A2 (en) | 2008-06-12 |
| ATE547394T1 (de) | 2012-03-15 |
| JP2014098008A (ja) | 2014-05-29 |
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