PL357928A1 - Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny - Google Patents

Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny

Info

Publication number
PL357928A1
PL357928A1 PL02357928A PL35792802A PL357928A1 PL 357928 A1 PL357928 A1 PL 357928A1 PL 02357928 A PL02357928 A PL 02357928A PL 35792802 A PL35792802 A PL 35792802A PL 357928 A1 PL357928 A1 PL 357928A1
Authority
PL
Poland
Prior art keywords
olanzapine
polymorphic form
pharmaceutically pure
pure polymorphic
obtaining pharmaceutically
Prior art date
Application number
PL02357928A
Other languages
English (en)
Other versions
PL202856B1 (pl
Inventor
Zbigniew Majka
Tomasz Stawiński
Original Assignee
ADAMED Sp.z o.o.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ADAMED Sp.z o.o. filed Critical ADAMED Sp.z o.o.
Priority to PL357928A priority Critical patent/PL202856B1/pl
Priority to CNB200380106963XA priority patent/CN100354280C/zh
Priority to BR0317594-4A priority patent/BR0317594A/pt
Priority to EP03768031A priority patent/EP1581537B1/en
Priority to CA002506663A priority patent/CA2506663A1/en
Priority to PCT/IB2003/005931 priority patent/WO2004056833A1/en
Priority to AU2003292452A priority patent/AU2003292452A1/en
Priority to HR20050549A priority patent/HRP20050549A2/hr
Priority to DE60317712T priority patent/DE60317712D1/de
Priority to UAA200507207A priority patent/UA82213C2/uk
Priority to ES03768031T priority patent/ES2294333T3/es
Priority to MXPA05006711A priority patent/MXPA05006711A/es
Publication of PL357928A1 publication Critical patent/PL357928A1/pl
Priority to NO20053368A priority patent/NO20053368L/no
Publication of PL202856B1 publication Critical patent/PL202856B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL357928A 2002-12-20 2002-12-20 Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny PL202856B1 (pl)

Priority Applications (13)

Application Number Priority Date Filing Date Title
PL357928A PL202856B1 (pl) 2002-12-20 2002-12-20 Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny
HR20050549A HRP20050549A2 (en) 2002-12-20 2003-12-15 A process for the preparation of a pharmaceutically pure polymorphic form i of olanzapine
DE60317712T DE60317712D1 (de) 2002-12-20 2003-12-15 Prozess zum Entfernen von Verunreinigung S von Olanzapin polymorpher Form I
EP03768031A EP1581537B1 (en) 2002-12-20 2003-12-15 Process for removing impurity S from olanzapine polymorphic form I
CA002506663A CA2506663A1 (en) 2002-12-20 2003-12-15 A process for the preparation of a pharmaceutically pure polymorphic form i of olanzapine
PCT/IB2003/005931 WO2004056833A1 (en) 2002-12-20 2003-12-15 A process for the preparation of a pharmaceutically pure polymorphic form i of olanzapine
AU2003292452A AU2003292452A1 (en) 2002-12-20 2003-12-15 A process for the preparation of a pharmaceutically pure polymorphic form i of olanzapine
CNB200380106963XA CN100354280C (zh) 2002-12-20 2003-12-15 一种制备药物纯奥氮平的多晶型ⅰ的方法
BR0317594-4A BR0317594A (pt) 2002-12-20 2003-12-15 Processo para a preparação de uma forma "i" de olanzapina polimórfica farmaceuticamente pura, produto resultante e processo para remoção da impureza "s" a partir da forma i polimórfica de olanzapina
UAA200507207A UA82213C2 (uk) 2002-12-20 2003-12-15 Спосіб очищення фармацевтично чистої поліморфної форми i оланзапіну
ES03768031T ES2294333T3 (es) 2002-12-20 2003-12-15 Procedimiento para la eliminacion de la impureza s de la forma polimorfica i de la olanzapina.
MXPA05006711A MXPA05006711A (es) 2002-12-20 2003-12-15 Un proceso para la preparacion de una forma i polimorfica farmaceuticamente pura de olanzapina.
NO20053368A NO20053368L (no) 2002-12-20 2005-07-11 Fremgangsmate for fremstilling av en farmasoytisk ren polymorf I av olanzapin.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PL357928A PL202856B1 (pl) 2002-12-20 2002-12-20 Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny

Publications (2)

Publication Number Publication Date
PL357928A1 true PL357928A1 (pl) 2004-06-28
PL202856B1 PL202856B1 (pl) 2009-07-31

Family

ID=32678125

Family Applications (1)

Application Number Title Priority Date Filing Date
PL357928A PL202856B1 (pl) 2002-12-20 2002-12-20 Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny

Country Status (13)

Country Link
EP (1) EP1581537B1 (pl)
CN (1) CN100354280C (pl)
AU (1) AU2003292452A1 (pl)
BR (1) BR0317594A (pl)
CA (1) CA2506663A1 (pl)
DE (1) DE60317712D1 (pl)
ES (1) ES2294333T3 (pl)
HR (1) HRP20050549A2 (pl)
MX (1) MXPA05006711A (pl)
NO (1) NO20053368L (pl)
PL (1) PL202856B1 (pl)
UA (1) UA82213C2 (pl)
WO (1) WO2004056833A1 (pl)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003300324A1 (en) 2002-12-24 2004-07-22 Teva Pharmaceutical Industries Ltd. Novel crystal forms of olanzapine, methods for their preparation and method for the preparation of known olanzapine crystal forms
WO2006025065A1 (en) * 2004-08-31 2006-03-09 Lee Pharma Private Limited A process for the preparation of anhydrous olanzopine hydrochloride of form-1
WO2006027800A1 (en) 2004-09-06 2006-03-16 Shasun Chemicals And Drugs Limited A novel process for preparation of a pharmaceutically pure polymorphic form 1 of olanzapine
GB0522473D0 (en) 2005-11-03 2005-12-14 Actavis Group A pharmaceutical formulation
WO2007144901A1 (en) * 2006-06-12 2007-12-21 Jubilant Organosys Limited Process for stabilization of olanzapine polymorphic form i
PL381564A1 (pl) 2007-01-22 2008-08-04 Koźluk Tomasz Nobilus Ent Sposób wytwarzania zasadniczo czystej odmiany polimorficznej I olanzapiny
EP2292624A1 (en) 2009-07-20 2011-03-09 LEK Pharmaceuticals d.d. Process for the purification of olanzapine
CN103910747B (zh) * 2014-04-24 2016-03-23 东南大学 一种奥氮平药物晶型f及其制备方法
CN109456336A (zh) * 2017-09-06 2019-03-12 万全万特制药江苏有限公司 奥氮平的精制方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5229382A (en) * 1990-04-25 1993-07-20 Lilly Industries Limited 2-methyl-thieno-benzodiazepine
GB9009229D0 (en) * 1990-04-25 1990-06-20 Lilly Industries Ltd Pharmaceutical compounds
EG23659A (en) * 1995-03-24 2007-03-26 Lilly Co Eli Process and crystal forms of methyl-thieno-benzodiazepine
CR5278A (es) * 1995-03-24 1996-07-04 Lilly Co Eli Formulacion oral de 2-metil-tieno-benzodiacepina
US5631250A (en) * 1995-03-24 1997-05-20 Eli Lilly And Company Process and solvate of 2-methyl-thieno-benzodiazepine
US6348458B1 (en) * 1999-12-28 2002-02-19 U & I Pharmaceuticals Ltd. Polymorphic forms of olanzapine
SK2502003A3 (en) * 2000-08-31 2004-03-02 Reddys Lab Ltd Dr Process for preparation of hydrates of olanzapine and their conversion into crystalline forms of olanzapine
PL196814B1 (pl) * 2002-05-17 2008-02-29 Inst Farmaceutyczny Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty
ATE500258T1 (de) * 2002-05-31 2011-03-15 Sandoz Ag Verfahren zur herstellung von olanzapin form i
SI21270A (sl) * 2002-07-15 2004-02-29 Krka, Tovarna Zdravil, D.D., Novo Mesto Kristalne oblike olanzapina in postopki za njihovo pripravo

Also Published As

Publication number Publication date
WO2004056833A1 (en) 2004-07-08
MXPA05006711A (es) 2005-11-23
NO20053368D0 (no) 2005-07-11
NO20053368L (no) 2005-07-11
BR0317594A (pt) 2005-11-22
EP1581537B1 (en) 2007-11-21
AU2003292452A1 (en) 2004-07-14
PL202856B1 (pl) 2009-07-31
ES2294333T3 (es) 2008-04-01
UA82213C2 (uk) 2008-03-25
CN100354280C (zh) 2007-12-12
HRP20050549A2 (en) 2005-12-31
CA2506663A1 (en) 2004-07-08
DE60317712D1 (de) 2008-01-03
EP1581537A1 (en) 2005-10-05
CN1729195A (zh) 2006-02-01

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