EG24142A - Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition - Google Patents

Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition

Info

Publication number
EG24142A
EG24142A EG20011058A EG20011058A EG24142A EG 24142 A EG24142 A EG 24142A EG 20011058 A EG20011058 A EG 20011058A EG 20011058 A EG20011058 A EG 20011058A EG 24142 A EG24142 A EG 24142A
Authority
EG
Egypt
Prior art keywords
preparing
preparation
pharmaceutical composition
crystalline monohydrate
monohydrate
Prior art date
Application number
EG20011058A
Other languages
English (en)
Inventor
Banholzer Rolf
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EG24142(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of EG24142A publication Critical patent/EG24142A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EG20011058A 2000-10-12 2001-10-09 Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition EG24142A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12

Publications (1)

Publication Number Publication Date
EG24142A true EG24142A (en) 2008-08-06

Family

ID=7659568

Family Applications (1)

Application Number Title Priority Date Filing Date
EG20011058A EG24142A (en) 2000-10-12 2001-10-09 Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition

Country Status (46)

Country Link
EP (2) EP1468998A1 (fr)
JP (1) JP3764422B2 (fr)
KR (1) KR100823860B1 (fr)
CN (2) CN100519558C (fr)
AP (1) AP1572A (fr)
AR (2) AR034389A1 (fr)
AT (1) ATE276253T1 (fr)
AU (2) AU2002214996B2 (fr)
BG (1) BG66161B1 (fr)
BR (1) BR0114584A (fr)
CA (1) CA2425539C (fr)
CR (1) CR6938A (fr)
CZ (1) CZ301841B6 (fr)
DE (1) DE50103666D1 (fr)
DK (1) DK1326862T3 (fr)
DZ (1) DZ3478A1 (fr)
EA (1) EA004381B1 (fr)
EC (1) ECSP034540A (fr)
EE (1) EE04567B1 (fr)
EG (1) EG24142A (fr)
ES (1) ES2228965T3 (fr)
GE (1) GEP20063905B (fr)
HR (1) HRP20030276B1 (fr)
HU (1) HU226830B1 (fr)
IL (2) IL155335A0 (fr)
IS (1) IS2339B (fr)
MA (1) MA25842A1 (fr)
ME (2) MEP40008A (fr)
MX (1) MXPA03003221A (fr)
MY (1) MY126931A (fr)
NO (1) NO328465B1 (fr)
NZ (1) NZ525733A (fr)
OA (1) OA12403A (fr)
PE (1) PE20020422A1 (fr)
PL (1) PL207870B1 (fr)
PT (1) PT1326862E (fr)
RS (1) RS50218B (fr)
SA (1) SA01220412B1 (fr)
SI (1) SI1326862T1 (fr)
SK (1) SK287009B6 (fr)
TR (1) TR200402579T4 (fr)
TW (1) TW589313B (fr)
UA (1) UA74215C2 (fr)
UY (2) UY26962A1 (fr)
WO (1) WO2002030928A1 (fr)
ZA (1) ZA200302500B (fr)

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DE10317461A1 (de) 2003-04-16 2004-10-28 Boehringer Ingelheim Pharma Gmbh & Co. Kg Radioaktiv markierte Mikropartikel, Verfahren zu deren Herstellung und deren Verwendung
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ES2523518T3 (es) 2004-04-22 2014-11-26 Boehringer Ingelheim International Gmbh Nuevas combinaciones farmacológicas para el tratamiento de enfermedades de las vías respiratorias
DE102004024454A1 (de) 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
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DE602004020337D1 (de) 2004-08-11 2009-05-14 Boehringer Ingelheim Pharma Anticholinergika enthaltende Arzneimittel zur Behandlung von Krankheiten der ableitenden Harnwege
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CN101163706A (zh) 2005-04-21 2008-04-16 贝林格尔·英格海姆国际有限公司 用于治疗炎性疾病的二氢噻吩并嘧啶
MX2007012907A (es) 2005-04-28 2008-03-14 Boehringer Ingelheim Int Nuevos compuestos para el tratamiento de enfermedades inflamatorias.
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EP2085396A3 (fr) 2005-05-02 2009-11-25 Boehringer Ingelheim International Gmbh Nouvelles formules cristallines de bromure de tiotropium
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CN101237872A (zh) * 2005-08-06 2008-08-06 贝林格尔·英格海姆国际有限公司 噻托铵盐在治疗严重持续性哮喘中的用途
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Also Published As

Publication number Publication date
SI1326862T1 (sl) 2005-02-28
PT1326862E (pt) 2004-11-30
AP2003002775A0 (en) 2003-03-31
UY34901A (es) 2015-02-27
CN1733761A (zh) 2006-02-15
EP1326862B1 (fr) 2004-09-15
EP1468998A1 (fr) 2004-10-20
IS6772A (is) 2003-04-09
PE20020422A1 (es) 2002-06-28
UY26962A1 (es) 2002-06-20
HRP20030276B1 (en) 2006-02-28
TW589313B (en) 2004-06-01
CR6938A (es) 2004-10-28
KR100823860B1 (ko) 2008-04-21
CZ301841B6 (cs) 2010-07-07
ES2228965T3 (es) 2005-04-16
BG107687A (bg) 2003-09-30
BR0114584A (pt) 2003-08-26
AU2002214996B2 (en) 2007-03-15
NO328465B1 (no) 2010-02-22
CN1469877A (zh) 2004-01-21
KR20030042008A (ko) 2003-05-27
MEP40008A (en) 2011-02-10
DE50103666D1 (de) 2004-10-21
ATE276253T1 (de) 2004-10-15
CA2425539C (fr) 2007-04-03
YU27303A (sh) 2006-05-25
HUP0301022A2 (hu) 2003-10-28
CN1221549C (zh) 2005-10-05
EE200300171A (et) 2003-06-16
HU226830B1 (en) 2009-11-30
ECSP034540A (es) 2003-07-25
HK1086557A1 (zh) 2006-09-22
ZA200302500B (en) 2004-04-22
DK1326862T3 (da) 2004-11-22
EA004381B1 (ru) 2004-04-29
NO20031694D0 (no) 2003-04-11
CA2425539A1 (fr) 2003-04-11
AU1499602A (en) 2002-04-22
NO20031694L (no) 2003-04-11
HK1060567A1 (en) 2004-08-13
CN100519558C (zh) 2009-07-29
EP1326862A1 (fr) 2003-07-16
IL155335A (en) 2009-02-11
AP1572A (en) 2006-02-13
IL155335A0 (en) 2003-11-23
GEP20063905B (en) 2006-08-25
SA01220412B1 (ar) 2006-11-05
MXPA03003221A (es) 2004-12-03
ME00243B (me) 2011-05-10
EE04567B1 (et) 2005-12-15
PL207870B1 (pl) 2011-02-28
RS50218B (sr) 2009-07-15
HUP0301022A3 (en) 2005-12-28
EA200300457A1 (ru) 2003-10-30
TR200402579T4 (tr) 2004-12-21
AR034389A1 (es) 2004-02-25
IS2339B (is) 2008-02-15
MY126931A (en) 2006-10-31
WO2002030928A1 (fr) 2002-04-18
UA74215C2 (uk) 2005-11-15
JP3764422B2 (ja) 2006-04-05
JP2004526668A (ja) 2004-09-02
BG66161B1 (bg) 2011-09-30
DZ3478A1 (fr) 2002-04-18
OA12403A (en) 2006-04-18
SK287009B6 (sk) 2009-09-07
AR068527A2 (es) 2009-11-18
MA25842A1 (fr) 2003-07-01
NZ525733A (en) 2005-01-28
PL366041A1 (en) 2005-01-24
HRP20030276A2 (en) 2005-02-28
SK4362003A3 (en) 2003-08-05

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