MA27069A1 - FORMES POLYMORPHES DE RIFAXIMIN, PROCEDES POUR LEUR PRODUCTION ET USAGE DE MeME DANS LES PREPARATIONS MEDICINALES - Google Patents

FORMES POLYMORPHES DE RIFAXIMIN, PROCEDES POUR LEUR PRODUCTION ET USAGE DE MeME DANS LES PREPARATIONS MEDICINALES

Info

Publication number
MA27069A1
MA27069A1 MA27590A MA27590A MA27069A1 MA 27069 A1 MA27069 A1 MA 27069A1 MA 27590 A MA27590 A MA 27590A MA 27590 A MA27590 A MA 27590A MA 27069 A1 MA27069 A1 MA 27069A1
Authority
MA
Morocco
Prior art keywords
rifaximin
production
medicinal preparations
crystallization
forms
Prior art date
Application number
MA27590A
Other languages
English (en)
Inventor
Giuseppe C Viscomi
Manuela Campana
Dario Braga
Donatella Confortini
Vincenzo Cannata
Denis Severini
Paolo Righi
Goffredo Rosini
Original Assignee
Alfa Wassermann Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33187382&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA27069(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alfa Wassermann Spa filed Critical Alfa Wassermann Spa
Publication of MA27069A1 publication Critical patent/MA27069A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • H—ELECTRICITY
    • H05—ELECTRIC TECHNIQUES NOT OTHERWISE PROVIDED FOR
    • H05B—ELECTRIC HEATING; ELECTRIC LIGHT SOURCES NOT OTHERWISE PROVIDED FOR; CIRCUIT ARRANGEMENTS FOR ELECTRIC LIGHT SOURCES, IN GENERAL
    • H05B6/00—Heating by electric, magnetic or electromagnetic fields
    • H05B6/02—Induction heating
    • H05B6/10—Induction heating apparatus, other than furnaces, for specific applications
    • H05B6/12—Cooking devices
    • H05B6/1209—Cooking devices induction cooking plates or the like and devices to be used in combination with them
    • H05B6/1236—Cooking devices induction cooking plates or the like and devices to be used in combination with them adapted to induce current in a coil to supply power to a device and electrical heating devices powered in this way
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • H—ELECTRICITY
    • H05—ELECTRIC TECHNIQUES NOT OTHERWISE PROVIDED FOR
    • H05B—ELECTRIC HEATING; ELECTRIC LIGHT SOURCES NOT OTHERWISE PROVIDED FOR; CIRCUIT ARRANGEMENTS FOR ELECTRIC LIGHT SOURCES, IN GENERAL
    • H05B6/00—Heating by electric, magnetic or electromagnetic fields
    • H05B6/02—Induction heating
    • H05B6/10—Induction heating apparatus, other than furnaces, for specific applications
    • H05B6/12—Cooking devices
    • H05B6/1209—Cooking devices induction cooking plates or the like and devices to be used in combination with them
    • H05B6/1245—Cooking devices induction cooking plates or the like and devices to be used in combination with them with special coil arrangements
    • H05B6/1263—Cooking devices induction cooking plates or the like and devices to be used in combination with them with special coil arrangements using coil cooling arrangements

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Physics & Mathematics (AREA)
  • Electromagnetism (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)

Abstract

FORMES POLYMORPHES DE RIFAXIMIN, PROCESSUS DE LEUR PRODUCTION ET DE LEUR EMPLOI DANS LES PREPARATIONS MEDICINALES Des formes cristallines polymorphes de l'antibiotique rifaximin (INN) dites rifaximin (alpha) et rifaximin (beta), et une forme faiblement cristalline appelée rifaximin (upsilon), ont été découvertes. Ces formes sont utiles dans la production des préparations médicinales pour l'usage oral et topique, et peuvent être obtenues au moyen d'un processus de cristallisation effectué par dissolvant chaud de rifaximin brute dans alcool de l'éthyle et en entraînant la cristallisation du produit par l'addition d'eau à une température déterminée pendant une période déterminée. La cristallisation est poursuivie par un séchage effectué sous des conditions contrôlées jusqu'à ce que le produit fini atteint une teneur d'eau spécifique.
MA27590A 2003-11-07 2004-03-24 FORMES POLYMORPHES DE RIFAXIMIN, PROCEDES POUR LEUR PRODUCTION ET USAGE DE MeME DANS LES PREPARATIONS MEDICINALES MA27069A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002144A ITMI20032144A1 (it) 2003-11-07 2003-11-07 Forme polimorfe di rifaximina, processi per ottenerle e

Publications (1)

Publication Number Publication Date
MA27069A1 true MA27069A1 (fr) 2004-12-20

Family

ID=33187382

Family Applications (1)

Application Number Title Priority Date Filing Date
MA27590A MA27069A1 (fr) 2003-11-07 2004-03-24 FORMES POLYMORPHES DE RIFAXIMIN, PROCEDES POUR LEUR PRODUCTION ET USAGE DE MeME DANS LES PREPARATIONS MEDICINALES

Country Status (37)

Country Link
US (5) US7045620B2 (fr)
EP (6) EP1676847B1 (fr)
JP (5) JP2005139161A (fr)
KR (4) KR20050043589A (fr)
CN (4) CN1613858A (fr)
AR (3) AR043547A1 (fr)
AT (3) ATE361927T1 (fr)
AU (2) AU2004200964A1 (fr)
BR (2) BRPI0402382A (fr)
CA (2) CA2460384A1 (fr)
CL (1) CL2004000498A1 (fr)
CO (1) CO5560083A1 (fr)
CY (3) CY1108017T1 (fr)
DE (4) DE602004019296D1 (fr)
DK (3) DK1557421T3 (fr)
ES (3) ES2244364T3 (fr)
HR (2) HRP20040265A2 (fr)
IL (2) IL160798A0 (fr)
IT (1) ITMI20032144A1 (fr)
JO (1) JO2470B1 (fr)
MA (1) MA27069A1 (fr)
MD (1) MD3653G8 (fr)
ME (1) ME00424B (fr)
MX (2) MXPA04002353A (fr)
NO (1) NO334950B1 (fr)
NZ (1) NZ531622A (fr)
PL (3) PL1557421T3 (fr)
PT (3) PT1557421E (fr)
RS (4) RS54571B1 (fr)
RU (1) RU2270200C2 (fr)
SI (3) SI1676848T1 (fr)
TN (2) TNSN04044A1 (fr)
TW (1) TWI285107B (fr)
UA (1) UA86384C2 (fr)
WO (1) WO2005044823A2 (fr)
YU (1) YU24804A (fr)
ZA (1) ZA200401948B (fr)

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WO2009108730A2 (fr) 2008-02-25 2009-09-03 Salix Pharmaceuticals, Ltd. Formes de rifaximine et utilisations correspondantes

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